A single point mutation in the seventh hydrophobic domain of the alpha 2-adrenergic receptor changes antagonist binding specificity to that of a beta receptor

Trans Assoc Am Physicians. 1991:104:62-8.
No abstract available

Publication types

  • Research Support, U.S. Gov't, P.H.S.
  • Review

MeSH terms

  • Adrenergic alpha-Antagonists / metabolism
  • Amino Acid Sequence
  • Animals
  • Binding Sites
  • Humans
  • Molecular Sequence Data
  • Point Mutation
  • Receptors, Adrenergic, alpha / genetics*
  • Receptors, Adrenergic, alpha / metabolism
  • Receptors, Adrenergic, beta / genetics
  • Receptors, Adrenergic, beta / metabolism

Substances

  • Adrenergic alpha-Antagonists
  • Receptors, Adrenergic, alpha
  • Receptors, Adrenergic, beta