Medicinal chemistry of hERG optimizations: Highlights and hang-ups

J Med Chem. 2006 Aug 24;49(17):5029-46. doi: 10.1021/jm060379l.
No abstract available

Publication types

  • Review

MeSH terms

  • Animals
  • Binding Sites
  • Chemistry, Pharmaceutical / methods
  • Ether-A-Go-Go Potassium Channels / antagonists & inhibitors
  • Ether-A-Go-Go Potassium Channels / chemistry*
  • Ether-A-Go-Go Potassium Channels / physiology
  • Humans
  • Molecular Structure
  • Potassium Channel Blockers / chemistry*
  • Potassium Channel Blockers / pharmacology
  • Structure-Activity Relationship

Substances

  • Ether-A-Go-Go Potassium Channels
  • Potassium Channel Blockers