Chronic benzodiazepine administration potentiates high voltage-activated calcium currents in hippocampal CA1 neurons

J Pharmacol Exp Ther. 2008 Dec;327(3):872-83. doi: 10.1124/jpet.108.144444. Epub 2008 Sep 23.

Abstract

Signs of physical dependence as a consequence of long-term drug use and a moderate abuse liability limit benzodiazepine clinical usefulness. Growing evidence suggests a role for voltage-gated calcium channel (VGCC) regulation in mediating a range of chronic drug effects from drug withdrawal phenomena to dependence on a variety of drugs of abuse. High voltage-activated (HVA) calcium currents were measured in whole-cell recordings from acutely isolated hippocampal CA1 neurons after a 1-week flurazepam (FZP) treatment that results in withdrawal-anxiety. An approximately 1.8-fold increase in Ca(2+) current density was detected immediately after and up to 2 days but not 3 or 4 days after drug withdrawal. Current density was unchanged after acute desalkyl-FZP treatment. A significant negative shift of the half-maximal potential of activation of HVA currents was also observed but steady-state inactivation remained unchanged. FZP and diazepam showed use- and concentration-dependent inhibition of Ca(2+) currents in hippocampal cultured cells following depolarizing trains (FZP, IC(50) = 1.8 microM; diazepam, IC(50) = 36 microM), pointing to an additional mechanism by which benzodiazepines modulate HVA Ca(2+) channels. Systemic preinjection of nimodipine (10 mg/kg), an L-type (L)-VGCC antagonist, prevented the benzodiazepine-induced increase in alpha-amino-3-hydroxy-5-methylisoxasole-4-propionic acid receptor (AMPAR)-mediated miniature excitatory postsynaptic current in CA1 neurons 2 days after FZP withdrawal, suggesting that AMPAR potentiation, previously linked to withdrawal-anxiety may require enhanced L-VGCC-mediated Ca(2+) influx. Taken together with prior work, these findings suggest that enhanced Ca(2+) entry through HVA Ca(2+) channels may contribute to hippocampal AMPAR plasticity and serve as a potential mechanism underlying benzodiazepine physical dependence.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Benzodiazepines / administration & dosage
  • Benzodiazepines / pharmacology*
  • Calcium / metabolism*
  • Calcium Channels / drug effects*
  • Calcium Channels / metabolism
  • Electrophysiology
  • Excitatory Postsynaptic Potentials / drug effects
  • Hippocampus / cytology*
  • Miniature Postsynaptic Potentials / drug effects
  • Pyramidal Cells / drug effects*
  • Pyramidal Cells / physiology
  • Rats
  • Receptors, Glutamate / physiology
  • Substance Withdrawal Syndrome
  • Substance-Related Disorders*

Substances

  • Calcium Channels
  • Receptors, Glutamate
  • Benzodiazepines
  • Calcium