Coibacins A and B: total synthesis and stereochemical revision

J Org Chem. 2014 Jan 17;79(2):630-42. doi: 10.1021/jo402339y. Epub 2014 Jan 9.

Abstract

The interface between synthetic organic chemistry and natural products was explored in order to unravel the structure of coibacin A, a metabolite isolated from the marine cyanobacterium cf. Oscillatoria sp. that exhibits selective antileishmanial activity and potent anti-inflammatory properties. Our synthetic plan focused on a convergent strategy that allows rapid access to the desired target by coupling of three key fragments involving E-selective Wittig and modified Julia olefinations. CD measurements and comparative HPLC analyses of the natural product and four synthetic stereoisomers led to determination of its absolute configuration, thus correcting the original assignment at C-5 and unambiguously establishing those at C-16 and C-18. Additionally, we synthesized coibacin B on the basis of the assignment of configuration for coibacin A.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Ketones / chemical synthesis*
  • Ketones / chemistry*
  • Ketones / isolation & purification
  • Lactones / chemical synthesis*
  • Lactones / chemistry*
  • Lactones / isolation & purification
  • Molecular Conformation
  • Oscillatoria / chemistry*
  • Stereoisomerism

Substances

  • Ketones
  • Lactones
  • coibacin A
  • coibacin B