The potential of targeting epigenetic regulators for the treatment of fibrotic cardiac diseases

Future Med Chem. 2016 Sep;8(13):1533-6. doi: 10.4155/fmc-2016-0144. Epub 2016 Aug 24.
No abstract available

Keywords: epigenetics; fibrosis; heart; small molecules.

Publication types

  • Editorial
  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Epigenomics*
  • Fibrosis
  • Heart Diseases / drug therapy
  • Heart Diseases / pathology*
  • Histone Deacetylase Inhibitors / chemistry
  • Histone Deacetylase Inhibitors / therapeutic use
  • Histone Deacetylases / chemistry
  • Histone Deacetylases / metabolism
  • Humans
  • Proteins / antagonists & inhibitors
  • Proteins / metabolism
  • RNA Polymerase II / metabolism
  • Small Molecule Libraries / chemistry
  • Small Molecule Libraries / therapeutic use

Substances

  • Histone Deacetylase Inhibitors
  • Proteins
  • Small Molecule Libraries
  • bromodomain and extra-terminal domain protein, human
  • RNA Polymerase II
  • Histone Deacetylases