Studies on the electrogenic action of acetylcholine with Torpedo marmorata electric organ. IV. Quinacrine: a fluorescent probe for the conformational transitions of the cholinergic receptor protein in its membrane-bound state

J Mol Biol. 1976 Sep 25;106(3):497-516. doi: 10.1016/0022-2836(76)90249-7.
No abstract available

MeSH terms

  • Acetylcholine / physiology*
  • Animals
  • Binding, Competitive
  • Carbachol / pharmacology
  • Cell Membrane / drug effects
  • Cell Membrane / physiology
  • Decamethonium Compounds / pharmacology
  • Electric Organ / physiology*
  • Fishes
  • Gallamine Triethiodide / pharmacology
  • Hexamethonium Compounds / pharmacology
  • Kinetics
  • Prilocaine / pharmacology
  • Protein Conformation
  • Quinacrine / pharmacology*
  • Receptors, Cholinergic / drug effects
  • Receptors, Cholinergic / physiology*
  • Spectrometry, Fluorescence

Substances

  • Decamethonium Compounds
  • Hexamethonium Compounds
  • Receptors, Cholinergic
  • Prilocaine
  • Carbachol
  • Quinacrine
  • Acetylcholine
  • Gallamine Triethiodide