Ber E - Search Results

1

Characterization of a novel, non-peptidyl antagonist of the human glucagon receptor.

Cascieri MA, Koch GE, Ber E, Sadowski SJ, Louizides D, de Laszlo SE, Hacker C, Hagmann WK, MacCoss M, Chicchi GG, Vicario PP. Cascieri MA, et al. Among authors: ber e. J Biol Chem. 1999 Mar 26;274(13):8694-7. doi: 10.1074/jbc.274.13.8694. J Biol Chem. 1999. PMID: 10085108 Free article.

2

Characterization of the binding of a potent, selective, radioiodinated antagonist to the human neurokinin-1 receptor.

Cascieri MA, Ber E, Fong TM, Sadowski S, Bansal A, Swain C, Seward E, Frances B, Burns D, Strader CD. Cascieri MA, et al. Among authors: ber e. Mol Pharmacol. 1992 Sep;42(3):458-63. Mol Pharmacol. 1992. PMID: 1383685

3

Purification and characterization of a unique, potent inhibitor of apamin binding from Leiurus quinquestriatus hebraeus venom.

Chicchi GG, Gimenez-Gallego G, Ber E, Garcia ML, Winquist R, Cascieri MA. Chicchi GG, et al. Among authors: ber e. J Biol Chem. 1988 Jul 25;263(21):10192-7. J Biol Chem. 1988. PMID: 2839478 Free article.

4

Characterization of the interaction of N-acyl-L-tryptophan benzyl ester neurokinin antagonists with the human neurokinin-1 receptor.

Cascieri MA, Macleod AM, Underwood D, Shiao LL, Ber E, Sadowski S, Yu H, Merchant KJ, Swain CJ, Strader CD, et al. Cascieri MA, et al. Among authors: ber e. J Biol Chem. 1994 Mar 4;269(9):6587-91. J Biol Chem. 1994. PMID: 7509807 Free article.

We have recently shown that a series of N-acyl-L-tryptophan benzyl esters are potent substance P antagonists (Macleod, A. M., Merchant, K. J., Cascieri, M. A., Sadowski, S., Ber, E., Swain, C. J., and Baker, R. (1993) J. Med Chem. 14, 2044-2045). ...

We have recently shown that a series of N-acyl-L-tryptophan benzyl esters are potent substance P antagonists (Macleod, A. M., Merchant, K. J …

5

Characterization of the interaction of diacylpiperazine antagonists with the human neurokinin-1 receptor: identification of a common binding site for structurally dissimilar antagonists.

Cascieri MA, Shiao LL, Mills SG, MacCoss M, Swain CJ, Yu H, Ber E, Sadowski S, Wu MT, Strader CD, et al. Cascieri MA, et al. Among authors: ber e. Mol Pharmacol. 1995 Apr;47(4):660-5. Mol Pharmacol. 1995. PMID: 7536886

6

Characterization of the binding and activity of a high affinity, pseudoirreversible morpholino tachykinin NK1 receptor antagonist.

Cascieri MA, Ber E, Fong TM, Hale JJ, Tang F, Shiao LL, Mills SG, MacCoss M, Sadowski S, Tota MR, Strader CD. Cascieri MA, et al. Among authors: ber e. Eur J Pharmacol. 1997 May 1;325(2-3):253-61. doi: 10.1016/s0014-2999(97)00122-2. Eur J Pharmacol. 1997. PMID: 9163573

7

Structural optimization affording 2-(R)-(1-(R)-3, 5-bis(trifluoromethyl)phenylethoxy)-3-(S)-(4-fluoro)phenyl-4- (3-oxo-1,2,4-triazol-5-yl)methylmorpholine, a potent, orally active, long-acting morpholine acetal human NK-1 receptor antagonist.

Hale JJ, Mills SG, MacCoss M, Finke PE, Cascieri MA, Sadowski S, Ber E, Chicchi GG, Kurtz M, Metzger J, Eiermann G, Tsou NN, Tattersall FD, Rupniak NM, Williams AR, Rycroft W, Hargreaves R, MacIntyre DE. Hale JJ, et al. Among authors: ber e. J Med Chem. 1998 Nov 5;41(23):4607-14. doi: 10.1021/jm980299k. J Med Chem. 1998. PMID: 9804700

8

Determination of the amino acid residues in substance P conferring selectivity and specificity for the rat neurokinin receptors.

Cascieri MA, Huang RR, Fong TM, Cheung AH, Sadowski S, Ber E, Strader CD. Cascieri MA, et al. Among authors: ber e. Mol Pharmacol. 1992 Jun;41(6):1096-9. Mol Pharmacol. 1992. PMID: 1377326

9

N-acyl-L-tryptophan benzyl esters: potent substance P receptor antagonists.

MacLeod AM, Merchant KJ, Cascieri MA, Sadowski S, Ber E, Swain CJ, Baker R. MacLeod AM, et al. Among authors: ber e. J Med Chem. 1993 Jul 9;36(14):2044-5. doi: 10.1021/jm00066a015. J Med Chem. 1993. PMID: 8393115 No abstract available.

10

Phosphorylated morpholine acetal human neurokinin-1 receptor antagonists as water-soluble prodrugs.

Hale JJ, Mills SG, MacCoss M, Dorn CP, Finke PE, Budhu RJ, Reamer RA, Huskey SE, Luffer-Atlas D, Dean BJ, McGowan EM, Feeney WP, Chiu SH, Cascieri MA, Chicchi GG, Kurtz MM, Sadowski S, Ber E, Tattersall FD, Rupniak NM, Williams AR, Rycroft W, Hargreaves R, Metzger JM, MacIntyre DE. Hale JJ, et al. Among authors: ber e. J Med Chem. 2000 Mar 23;43(6):1234-41. doi: 10.1021/jm990617v. J Med Chem. 2000. PMID: 10737756

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