Souers A - Search Results

1

Compounds that activate the mouse melanocortin-1 receptor identified by screening a small molecule library based upon the beta-turn.

Haskell-Luevano C, Rosenquist A, Souers A, Khong KC, Ellman JA, Cone RD. Haskell-Luevano C, et al. Among authors: souers a. J Med Chem. 1999 Oct 21;42(21):4380-7. doi: 10.1021/jm990190s. J Med Chem. 1999. PMID: 10543881

2

Novel inhibitors of alpha 4 beta 1 integrin receptor interactions through library synthesis and screening.

Souers AJ, Virgilio AA, Schürer SS, Ellman JA, Kogan TP, West HE, Ankener W, Vanderslice P. Souers AJ, et al. Bioorg Med Chem Lett. 1998 Sep 8;8(17):2297-302. doi: 10.1016/s0960-894x(98)00416-8. Bioorg Med Chem Lett. 1998. PMID: 9873531

3

Optimization of a somatostatin mimetic via constrained amino acid and backbone incorporation.

Souers AJ, Rosenquist A, Jarvie EM, Ladlow M, Feniuk W, Ellman JA. Souers AJ, et al. Bioorg Med Chem Lett. 2000 Dec 18;10(24):2731-3. doi: 10.1016/s0960-894x(00)00552-7. Bioorg Med Chem Lett. 2000. PMID: 11133079

4

Asymmetric synthesis of a C-3 substituted pipecolic acid.

Souers AJ, Ellman JA. Souers AJ, et al. J Org Chem. 2000 Feb 25;65(4):1222-4. doi: 10.1021/jo991293l. J Org Chem. 2000. PMID: 10814077 No abstract available.

5

The preparation and utility of bis(sulfinyl)imidoamidine ligands for the copper-catalyzed Diels-Alder reaction.

Owens TD, Souers AJ, Ellman JA. Owens TD, et al. Among authors: souers aj. J Org Chem. 2003 Jan 10;68(1):3-10. doi: 10.1021/jo020524c. J Org Chem. 2003. PMID: 12515453

6

Synthesis and crystal structure of a unique and homochiral N,S-bonded N,N'-bis(tert-butanesulfinyl)amidinate rhodium(I) complex.

Souers AJ, Owens TD, Oliver AG, Hollander FJ, Ellman JA. Souers AJ, et al. Inorg Chem. 2001 Sep 24;40(20):5299-301. doi: 10.1021/ic0104205. Inorg Chem. 2001. PMID: 11559098 No abstract available.

7

Microwave-assisted C-H bond activation: a rapid entry into functionalized heterocycles.

Tan KL, Vasudevan A, Bergman RG, Ellman JA, Souers AJ. Tan KL, et al. Among authors: souers aj. Org Lett. 2003 Jun 12;5(12):2131-4. doi: 10.1021/ol030050j. Org Lett. 2003. PMID: 12790546

8

Quinazoline sulfonamides as dual binders of the proteins B-cell lymphoma 2 and B-cell lymphoma extra long with potent proapoptotic cell-based activity.

Sleebs BE, Czabotar PE, Fairbrother WJ, Fairlie WD, Flygare JA, Huang DC, Kersten WJ, Koehler MF, Lessene G, Lowes K, Parisot JP, Smith BJ, Smith ML, Souers AJ, Street IP, Yang H, Baell JB. Sleebs BE, et al. Among authors: souers aj. J Med Chem. 2011 Mar 24;54(6):1914-26. doi: 10.1021/jm101596e. Epub 2011 Mar 2. J Med Chem. 2011. PMID: 21366295

9

Synthesis and evaluation of urea-based indazoles as melanin-concentrating hormone receptor 1 antagonists for the treatment of obesity.

Souers AJ, Gao J, Wodka D, Judd AS, Mulhern MM, Napier JJ, Brune ME, Bush EN, Brodjian SJ, Dayton BD, Shapiro R, Hernandez LE, Marsh KC, Sham HL, Collins CA, Kym PR. Souers AJ, et al. Bioorg Med Chem Lett. 2005 Jun 2;15(11):2752-7. doi: 10.1016/j.bmcl.2005.03.114. Bioorg Med Chem Lett. 2005. PMID: 15911251

10

Screening for cardiovascular safety: a structure-activity approach for guiding lead selection of melanin concentrating hormone receptor 1 antagonists.

Kym PR, Souers AJ, Campbell TJ, Lynch JK, Judd AS, Iyengar R, Vasudevan A, Gao J, Freeman JC, Wodka D, Mulhern M, Zhao G, Wagaw SH, Napier JJ, Brodjian S, Dayton BD, Reilly RM, Segreti JA, Fryer RM, Preusser LC, Reinhart GA, Hernandez L, Marsh KC, Sham HL, Collins CA, Polakowski JS. Kym PR, et al. Among authors: souers aj. J Med Chem. 2006 Apr 6;49(7):2339-52. doi: 10.1021/jm0512286. J Med Chem. 2006. PMID: 16570930

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