Search Page
Save citations to file
Email citations
Send citations to clipboard
Add to Collections
Add to My Bibliography
Create a file for external citation management software
Your saved search
Your RSS Feed
Search Results
8 results
Filters applied: . Clear all
Results are displayed in a computed author sort order.
The Results By Year timeline is not available.
Page 1
Design and development of selective muscarinic agonists for the treatment of Alzheimer's disease: characterization of tetrahydropyrimidine derivatives and development of new approaches for improved affinity and selectivity for M1 receptors.
Pharm Acta Helv. 2000 Mar;74(2-3):135-40. doi: 10.1016/s0031-6865(99)00026-6.
Pharm Acta Helv. 2000.
PMID: 10812950
Synthesis and biochemical activity of novel amidine derivatives as m1 muscarinic receptor agonists.
Ojo B, Dunbar PG, Durant GJ, Nagy PI, Huzl JJ 3rd, Periyasamy S, Ngur DO, el-Assadi AA, Hoss WP, Messer WS Jr.
Ojo B, et al. Among authors: el assadi aa.
Bioorg Med Chem. 1996 Oct;4(10):1605-15. doi: 10.1016/0968-0896(96)00152-6.
Bioorg Med Chem. 1996.
PMID: 8931930
Item in Clipboard
Synthesis and biological characterization of 1,4,5,6-tetrahydropyrimidine and 2-amino-3,4,5,6-tetrahydropyridine derivatives as selective m1 agonists.
Messer WS Jr, Abuh YF, Liu Y, Periyasamy S, Ngur DO, Edgar MA, El-Assadi AA, Sbeih S, Dunbar PG, Roknich S, Rho T, Fang Z, Ojo B, Zhang H, Huzl JJ 3rd, Nagy PI.
Messer WS Jr, et al. Among authors: el assadi aa.
J Med Chem. 1997 Apr 11;40(8):1230-46. doi: 10.1021/jm960467d.
J Med Chem. 1997.
PMID: 9111297
Item in Clipboard
Design, synthesis, and neurochemical evaluation of 5-(3-alkyl-1,2,4- oxadiazol-5-yl)-1,4,5,6-tetrahydropyrimidines as M1 muscarinic receptor agonists.
Dunbar PG, Durant GJ, Fang Z, Abuh YF, el-Assadi AA, Ngur DO, Periyasamy S, Hoss WP, Messer WS Jr.
Dunbar PG, et al. Among authors: el assadi aa.
J Med Chem. 1993 Apr 2;36(7):842-7. doi: 10.1021/jm00059a008.
J Med Chem. 1993.
PMID: 8464038
Item in Clipboard
Design, synthesis, and neurochemical evaluation of 2-amino-5-(alkoxycarbonyl)-3,4,5,6-tetrahydropyridines and 2-amino-5-(alkoxycarbonyl)-1,4,5,6-tetrahydropyrimidines as M1 muscarinic receptor agonists.
Dunbar PG, Durant GJ, Rho T, Ojo B, Huzl JJ 3rd, Smith DA, el-Assadi AA, Sbeih S, Ngur DO, Periyasamy S, et al.
Dunbar PG, et al. Among authors: el assadi aa.
J Med Chem. 1994 Aug 19;37(17):2774-82. doi: 10.1021/jm00043a016.
J Med Chem. 1994.
PMID: 8064804
Item in Clipboard
Synthesis and CLOGP correlation of imidooxy anticonvulsants.
Farrar VA, Ciechanowicz-Rutkowska M, Grochowski J, Serda P, Pilati T, Filippini G, Hinko CN, el-Assadi A, Moore JA, Edafiogho IO, et al.
Farrar VA, et al.
J Med Chem. 1993 Nov 12;36(23):3517-25. doi: 10.1021/jm00075a005.
J Med Chem. 1993.
PMID: 8246220
Item in Clipboard
Synthesis and anticonvulsant activity of enaminones. 2. Further structure-activity correlations.
Scott KR, Edafiogho IO, Richardson EL, Farrar VA, Moore JA, Tietz EI, Hinko CN, Chang H, el-Assadi A, Nicholson JM.
Scott KR, et al.
J Med Chem. 1993 Jul 9;36(14):1947-55. doi: 10.1021/jm00066a003.
J Med Chem. 1993.
PMID: 8336334
Item in Clipboard
Anticonvulsant activity of novel derivatives of 2- and 3-piperidinecarboxylic acid in mice and rats.
Hinko CN, Crider AM, Kliem MA, Steinmiller CL, Seo TH, Ho B, Venkatarangan P, el-Assadi AA, Chang H, Burns CM, Tietz EI, Andersen PH, Klitgaard H.
Hinko CN, et al. Among authors: el assadi aa.
Neuropharmacology. 1996;35(12):1721-35. doi: 10.1016/s0028-3908(96)00105-0.
Neuropharmacology. 1996.
PMID: 9076751
Item in Clipboard
Cite
Cite