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Structurally simplified macrolactone analogues of halichondrin B.
Bioorg Med Chem Lett. 2004 Nov 15;14(22):5547-50. doi: 10.1016/j.bmcl.2004.08.068.
Bioorg Med Chem Lett. 2004.
PMID: 15482921
Macrocyclic ketone analogues of halichondrin B.
Zheng W, Seletsky BM, Palme MH, Lydon PJ, Singer LA, Chase CE, Lemelin CA, Shen Y, Davis H, Tremblay L, Towle MJ, Salvato KA, Wels BF, Aalfs KK, Kishi Y, Littlefield BA, Yu MJ.
Zheng W, et al. Among authors: aalfs kk.
Bioorg Med Chem Lett. 2004 Nov 15;14(22):5551-4. doi: 10.1016/j.bmcl.2004.08.069.
Bioorg Med Chem Lett. 2004.
PMID: 15482922
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In vitro and in vivo anticancer activities of synthetic macrocyclic ketone analogues of halichondrin B.
Towle MJ, Salvato KA, Budrow J, Wels BF, Kuznetsov G, Aalfs KK, Welsh S, Zheng W, Seletsky BM, Palme MH, Habgood GJ, Singer LA, Dipietro LV, Wang Y, Chen JJ, Quincy DA, Davis A, Yoshimatsu K, Kishi Y, Yu MJ, Littlefield BA.
Towle MJ, et al. Among authors: aalfs kk.
Cancer Res. 2001 Feb 1;61(3):1013-21.
Cancer Res. 2001.
PMID: 11221827
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Eribulin induces irreversible mitotic blockade: implications of cell-based pharmacodynamics for in vivo efficacy under intermittent dosing conditions.
Towle MJ, Salvato KA, Wels BF, Aalfs KK, Zheng W, Seletsky BM, Zhu X, Lewis BM, Kishi Y, Yu MJ, Littlefield BA.
Towle MJ, et al. Among authors: aalfs kk.
Cancer Res. 2011 Jan 15;71(2):496-505. doi: 10.1158/0008-5472.CAN-10-1874. Epub 2010 Dec 2.
Cancer Res. 2011.
PMID: 21127197
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Covalent binding of 7,12-dimethylbenz(a)anthracene and 10-fluoro-7,12-dimethylbenz(a)anthracene to mouse epidermal DNA and its relationship to tumor-initiating activity.
DiGiovanni J, Fisher EP, Aalfs KK, Prichett WP.
DiGiovanni J, et al. Among authors: aalfs kk.
Cancer Res. 1985 Feb;45(2):591-7.
Cancer Res. 1985.
PMID: 3917851
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Mechanism of mouse skin tumor promotion by chrysarobin.
DiGiovanni J, Decina PC, Prichett WP, Cantor J, Aalfs KK, Coombs MM.
DiGiovanni J, et al. Among authors: aalfs kk.
Cancer Res. 1985 Jun;45(6):2584-9.
Cancer Res. 1985.
PMID: 3986797
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Formation and disappearance of benzo[a]pyrene DNA-adducts in mouse epidermis.
DiGiovanni J, Decina PC, Prichett WP, Fisher EP, Aalfs KK.
DiGiovanni J, et al. Among authors: aalfs kk.
Carcinogenesis. 1985 May;6(5):741-7. doi: 10.1093/carcin/6.5.741.
Carcinogenesis. 1985.
PMID: 3924430
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