Grabowski EJ - Search Results

1

Practical asymmetric synthesis of a potent PDE4 inhibitor via stereoselective enolate alkylation of a chiral aryl-heteroaryl secondary tosylate.

O'Shea PD, Chen CY, Chen W, Dagneau P, Frey LF, Grabowski EJ, Marcantonio KM, Reamer RA, Tan L, Tillyer RD, Roy A, Wang X, Zhao D. O'Shea PD, et al. Among authors: grabowski ej. J Org Chem. 2005 Apr 15;70(8):3021-30. doi: 10.1021/jo048156v. J Org Chem. 2005. PMID: 15822960

2

Practical asymmetric synthesis of a potent Cathepsin K inhibitor. Efficient palladium removal following Suzuki coupling.

Chen CY, Dagneau P, Grabowski EJ, Oballa R, O'Shea P, Prasit P, Robichaud J, Tillyer R, Wang X. Chen CY, et al. Among authors: grabowski ej. J Org Chem. 2003 Apr 4;68(7):2633-8. doi: 10.1021/jo0205614. J Org Chem. 2003. PMID: 12662032

3

Practical synthesis of a potent hepatitis C virus RNA replication inhibitor.

Bio MM, Xu F, Waters M, Williams JM, Savary KA, Cowden CJ, Yang C, Buck E, Song ZJ, Tschaen DM, Volante RP, Reamer RA, Grabowski EJ. Bio MM, et al. Among authors: grabowski ej. J Org Chem. 2004 Sep 17;69(19):6257-66. doi: 10.1021/jo0491096. J Org Chem. 2004. PMID: 15357584

4

Asymmetric synthesis of a prostaglandin D2 receptor antagonist.

Campos KR, Journet M, Lee S, Grabowski EJ, Tillyer RD. Campos KR, et al. Among authors: grabowski ej. J Org Chem. 2005 Jan 7;70(1):268-74. doi: 10.1021/jo048305+. J Org Chem. 2005. PMID: 15624932

5

Stereoselective formation of carbon-carbon bonds via SN2-displacement: synthesis of substituted cycloalkyl[b]indoles.

Hillier MC, Marcoux JF, Zhao D, Grabowski EJ, McKeown AE, Tillyer RD. Hillier MC, et al. Among authors: grabowski ej. J Org Chem. 2005 Oct 14;70(21):8385-94. doi: 10.1021/jo051146p. J Org Chem. 2005. PMID: 16209582

6

Highly Chemoselective Trichloroacetimidate-Mediated Alkylation of Ascomycin: A Convergent, Practical Synthesis of the Immunosuppressant L-733,725.

Song Z, DeMarco A, Zhao M, Corley EG, Thompson AS, McNamara J, Li Y, Rieger D, Sohar P, Mathre DJ, Tschaen DM, Reamer RA, Huntington MF, Ho GJ, Tsay FR, Emerson K, Shuman R, Grabowski EJ, Reider PJ. Song Z, et al. Among authors: grabowski ej. J Org Chem. 1999 Mar 19;64(6):1859-1867. doi: 10.1021/jo981805g. J Org Chem. 1999. PMID: 11674275

7

Synthesis of substituted imidazoles via organocatalysis.

Frantz DE, Morency L, Soheili A, Murry JA, Grabowski EJ, Tillyer RD. Frantz DE, et al. Among authors: grabowski ej. Org Lett. 2004 Mar 4;6(5):843-6. doi: 10.1021/ol0498803. Org Lett. 2004. PMID: 14986989

8

Practical asymmetric synthesis of a selective endothelin A receptor (ETA) antagonist.

Song ZJ, Zhao M, Frey L, Li J, Tan L, Chen CY, Tschaen DM, Tillyer R, Grabowski EJ, Volante R, Reider PJ, Kato Y, Okada S, Nemoto T, Sato H, Akao A, Mase T. Song ZJ, et al. Among authors: grabowski ej. Org Lett. 2001 Oct 18;3(21):3357-60. doi: 10.1021/ol016601s. Org Lett. 2001. PMID: 11594833

9

A Novel, Highly Enantioselective Ketone Alkynylation Reaction Mediated by Chiral Zinc Aminoalkoxides.

Tan L, Chen CY, Tillyer RD, Grabowski EJJ, Reider PJ. Tan L, et al. Angew Chem Int Ed Engl. 1999 Mar 1;38(5):711-713. doi: 10.1002/(SICI)1521-3773(19990301)38:5<711::AID-ANIE711>3.0.CO;2-W. Angew Chem Int Ed Engl. 1999. PMID: 29711532

10

Highly efficient synthesis of beta-amino acid derivatives via asymmetric hydrogenation of unprotected enamines.

Hsiao Y, Rivera NR, Rosner T, Krska SW, Njolito E, Wang F, Sun Y, Armstrong JD 3rd, Grabowski EJ, Tillyer RD, Spindler F, Malan C. Hsiao Y, et al. Among authors: grabowski ej. J Am Chem Soc. 2004 Aug 18;126(32):9918-9. doi: 10.1021/ja047901i. J Am Chem Soc. 2004. PMID: 15303855

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