Tillyer RD - Search Results

1

Practical asymmetric synthesis of a potent PDE4 inhibitor via stereoselective enolate alkylation of a chiral aryl-heteroaryl secondary tosylate.

O'Shea PD, Chen CY, Chen W, Dagneau P, Frey LF, Grabowski EJ, Marcantonio KM, Reamer RA, Tan L, Tillyer RD, Roy A, Wang X, Zhao D. O'Shea PD, et al. Among authors: tillyer rd. J Org Chem. 2005 Apr 15;70(8):3021-30. doi: 10.1021/jo048156v. J Org Chem. 2005. PMID: 15822960

2

Asymmetric synthesis of a prostaglandin D2 receptor antagonist.

Campos KR, Journet M, Lee S, Grabowski EJ, Tillyer RD. Campos KR, et al. Among authors: tillyer rd. J Org Chem. 2005 Jan 7;70(1):268-74. doi: 10.1021/jo048305+. J Org Chem. 2005. PMID: 15624932

3

Stereoselective formation of carbon-carbon bonds via SN2-displacement: synthesis of substituted cycloalkyl[b]indoles.

Hillier MC, Marcoux JF, Zhao D, Grabowski EJ, McKeown AE, Tillyer RD. Hillier MC, et al. Among authors: tillyer rd. J Org Chem. 2005 Oct 14;70(21):8385-94. doi: 10.1021/jo051146p. J Org Chem. 2005. PMID: 16209582

4

Nucleophilic displacement at benzhydryl centers: asymmetric synthesis of 1,1-diarylalkyl derivatives.

Bolshan Y, Chen CY, Chilenski JR, Gosselin F, Mathre DJ, O'Shea PD, Roy A, Tillyer RD. Bolshan Y, et al. Among authors: tillyer rd. Org Lett. 2004 Jan 8;6(1):111-4. doi: 10.1021/ol0361655. Org Lett. 2004. PMID: 14703363

5

Practical asymmetric synthesis of a potent Cathepsin K inhibitor. Efficient palladium removal following Suzuki coupling.

Chen CY, Dagneau P, Grabowski EJ, Oballa R, O'Shea P, Prasit P, Robichaud J, Tillyer R, Wang X. Chen CY, et al. J Org Chem. 2003 Apr 4;68(7):2633-8. doi: 10.1021/jo0205614. J Org Chem. 2003. PMID: 12662032

6

Practical asymmetric synthesis of a selective endothelin A receptor (ETA) antagonist.

Song ZJ, Zhao M, Frey L, Li J, Tan L, Chen CY, Tschaen DM, Tillyer R, Grabowski EJ, Volante R, Reider PJ, Kato Y, Okada S, Nemoto T, Sato H, Akao A, Mase T. Song ZJ, et al. Org Lett. 2001 Oct 18;3(21):3357-60. doi: 10.1021/ol016601s. Org Lett. 2001. PMID: 11594833

7

Synthesis of substituted imidazoles via organocatalysis.

Frantz DE, Morency L, Soheili A, Murry JA, Grabowski EJ, Tillyer RD. Frantz DE, et al. Among authors: tillyer rd. Org Lett. 2004 Mar 4;6(5):843-6. doi: 10.1021/ol0498803. Org Lett. 2004. PMID: 14986989

8

Stereoselective syntheses of highly functionalized bicyclo[3.1.0]hexanes: a general methodology for the synthesis of potent and selective mGluR2/3 agonists.

Tan L, Yasuda N, Yoshikawa N, Hartner FW, Eng KK, Leonard WR, Tsay FR, Volante RP, Tillyer RD. Tan L, et al. Among authors: tillyer rd. J Org Chem. 2005 Sep 30;70(20):8027-34. doi: 10.1021/jo0511187. J Org Chem. 2005. PMID: 16277324

9

An efficient asymmetric synthesis of an estrogen receptor modulator by sulfoxide-directed borane reduction.

Song ZJ, King AO, Waters MS, Lang F, Zewge D, Bio M, Leazer JL Jr, Javadi G, Kassim A, Tschaen DM, Reamer RA, Rosner T, Chilenski JR, Mathre DJ, Volante RP, Tillyer R. Song ZJ, et al. Proc Natl Acad Sci U S A. 2004 Apr 20;101(16):5776-81. doi: 10.1073/pnas.0307415101. Epub 2004 Apr 12. Proc Natl Acad Sci U S A. 2004. PMID: 15079059 Free PMC article.

10

Highly efficient synthesis of beta-amino acid derivatives via asymmetric hydrogenation of unprotected enamines.

Hsiao Y, Rivera NR, Rosner T, Krska SW, Njolito E, Wang F, Sun Y, Armstrong JD 3rd, Grabowski EJ, Tillyer RD, Spindler F, Malan C. Hsiao Y, et al. Among authors: tillyer rd. J Am Chem Soc. 2004 Aug 18;126(32):9918-9. doi: 10.1021/ja047901i. J Am Chem Soc. 2004. PMID: 15303855

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