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SM16, an orally active TGF-beta type I receptor inhibitor prevents myofibroblast induction and vascular fibrosis in the rat carotid injury model.
Arterioscler Thromb Vasc Biol. 2008 Apr;28(4):665-71. doi: 10.1161/ATVBAHA.107.158030. Epub 2008 Jan 17.
Arterioscler Thromb Vasc Biol. 2008.
PMID: 18202322
Potent and orally bioavailable 8-bicyclo[2.2.2]octylxanthines as adenosine A1 receptor antagonists.
Kiesman WF, Zhao J, Conlon PR, Dowling JE, Petter RC, Lutterodt F, Jin X, Smits G, Fure M, Jayaraj A, Kim J, Sullivan G, Linden J.
Kiesman WF, et al. Among authors: lutterodt f.
J Med Chem. 2006 Nov 30;49(24):7119-31. doi: 10.1021/jm0605381.
J Med Chem. 2006.
PMID: 17125264
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Tricyclic imidazoline derivatives as potent and selective adenosine A1 receptor antagonists.
Vu CB, Kiesman WF, Conlon PR, Lin KC, Tam M, Petter RC, Smits G, Lutterodt F, Jin X, Chen L, Zhang J.
Vu CB, et al. Among authors: lutterodt f.
J Med Chem. 2006 Nov 30;49(24):7132-9. doi: 10.1021/jm060539t.
J Med Chem. 2006.
PMID: 17125265
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Norbornyllactone-substituted xanthines as adenosine A(1) receptor antagonists.
Kiesman WF, Zhao J, Conlon PR, Petter RC, Jin X, Smits G, Lutterodt F, Sullivan GW, Linden J.
Kiesman WF, et al. Among authors: lutterodt f.
Bioorg Med Chem. 2006 Jun 1;14(11):3654-61. doi: 10.1016/j.bmc.2006.01.021. Epub 2006 Feb 2.
Bioorg Med Chem. 2006.
PMID: 16458010
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