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7 results
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Discovery of a potent, metabolically stabilized resorcylic lactone as an anti-inflammatory lead.
Bioorg Med Chem Lett. 2009 Nov 1;19(21):6196-9. doi: 10.1016/j.bmcl.2009.08.096. Epub 2009 Sep 3.
Bioorg Med Chem Lett. 2009.
PMID: 19783437
Discovery of anti-inflammatory clinical candidate E6201, inspired from resorcylic lactone LL-Z1640-2, III.
Shen Y, Boivin R, Yoneda N, Du H, Schiller S, Matsushima T, Goto M, Shirota H, Gusovsky F, Lemelin C, Jiang Y, Zhang Z, Pelletier R, Ikemori-Kawada M, Kawakami Y, Inoue A, Schnaderbeck M, Wang Y.
Shen Y, et al. Among authors: ikemori kawada m.
Bioorg Med Chem Lett. 2010 May 15;20(10):3155-7. doi: 10.1016/j.bmcl.2010.03.087. Epub 2010 Mar 30.
Bioorg Med Chem Lett. 2010.
PMID: 20399648
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Discovery of an in vitro and in vivo potent resorcylic lactone analog of LL-Z1640-2 as anti-inflammatory lead, II.
Shen Y, Du H, Kotake M, Matsushima T, Goto M, Shirota H, Gusovsky F, Li X, Jiang Y, Schiller S, Spyvee M, Davis H, Zhang Z, Pelletier R, Ikemori-Kawada M, Kawakami Y, Inoue A, Wang Y.
Shen Y, et al. Among authors: ikemori kawada m.
Bioorg Med Chem Lett. 2010 May 15;20(10):3047-9. doi: 10.1016/j.bmcl.2010.03.119. Epub 2010 Apr 9.
Bioorg Med Chem Lett. 2010.
PMID: 20427182
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Conformational analyses and MO studies of f152A1 and its analogues as potent protein kinase inhibitors.
Ikemori-Kawada M, Kawai T, Goto M, Wang YJ, Kawakami Y.
Ikemori-Kawada M, et al.
J Chem Inf Model. 2009 Dec;49(12):2650-9. doi: 10.1021/ci9003128.
J Chem Inf Model. 2009.
PMID: 19995092
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Docking simulation study and kinase selectivity of f152A1 and its analogs.
Ikemori-Kawada M, Inoue A, Goto M, Wang YJ, Kawakami Y.
Ikemori-Kawada M, et al.
J Chem Inf Model. 2012 Aug 27;52(8):2059-68. doi: 10.1021/ci300135g. Epub 2012 Aug 9.
J Chem Inf Model. 2012.
PMID: 22830536
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Distinct binding mode of multikinase inhibitor lenvatinib revealed by biochemical characterization.
Okamoto K, Ikemori-Kawada M, Jestel A, von König K, Funahashi Y, Matsushima T, Tsuruoka A, Inoue A, Matsui J.
Okamoto K, et al. Among authors: ikemori kawada m.
ACS Med Chem Lett. 2014 Nov 17;6(1):89-94. doi: 10.1021/ml500394m. eCollection 2015 Jan 8.
ACS Med Chem Lett. 2014.
PMID: 25589937
Free PMC article.
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Lenvatinib inhibits angiogenesis and tumor fibroblast growth factor signaling pathways in human hepatocellular carcinoma models.
Matsuki M, Hoshi T, Yamamoto Y, Ikemori-Kawada M, Minoshima Y, Funahashi Y, Matsui J.
Matsuki M, et al. Among authors: ikemori kawada m.
Cancer Med. 2018 Jun;7(6):2641-2653. doi: 10.1002/cam4.1517. Epub 2018 May 7.
Cancer Med. 2018.
PMID: 29733511
Free PMC article.
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