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Stereochemistry-activity relationship of orally active tetralin S1P agonist prodrugs.
Bioorg Med Chem Lett. 2010 Apr 1;20(7):2264-9. doi: 10.1016/j.bmcl.2010.02.006. Epub 2010 Feb 6.
Bioorg Med Chem Lett. 2010.
PMID: 20188554
Free PMC article.
Piperazine derivatives of [1,2,4]triazolo[1,5-a][1,3,5]triazine as potent and selective adenosine A2a receptor antagonists.
Vu CB, Peng B, Kumaravel G, Smits G, Jin X, Phadke D, Engber T, Huang C, Reilly J, Tam S, Grant D, Hetu G, Chen L, Zhang J, Petter RC.
Vu CB, et al. Among authors: hetu g.
J Med Chem. 2004 Aug 12;47(17):4291-9. doi: 10.1021/jm0498405.
J Med Chem. 2004.
PMID: 15294001
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2-Aminoimidazoles inhibitors of TGF-beta receptor 1.
Bonafoux D, Chuaqui C, Boriack-Sjodin PA, Fitch C, Hankins G, Josiah S, Black C, Hetu G, Ling L, Lee WC.
Bonafoux D, et al. Among authors: hetu g.
Bioorg Med Chem Lett. 2009 Feb 1;19(3):912-6. doi: 10.1016/j.bmcl.2008.11.119. Epub 2008 Dec 11.
Bioorg Med Chem Lett. 2009.
PMID: 19135364
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Novel diamino derivatives of [1,2,4]triazolo[1,5-a][1,3,5]triazine as potent and selective adenosine A2a receptor antagonists.
Vu CB, Pan D, Peng B, Kumaravel G, Smits G, Jin X, Phadke D, Engber T, Huang C, Reilly J, Tam S, Grant D, Hetu G, Petter RC.
Vu CB, et al. Among authors: hetu g.
J Med Chem. 2005 Mar 24;48(6):2009-18. doi: 10.1021/jm0498396.
J Med Chem. 2005.
PMID: 15771443
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Cerebrospinal fluid can be used as a surrogate to assess brain exposures of breast cancer resistance protein and P-glycoprotein substrates.
Xiao G, Black C, Hetu G, Sands E, Wang J, Caputo R, Rohde E, Gan LS.
Xiao G, et al. Among authors: hetu g.
Drug Metab Dispos. 2012 Apr;40(4):779-87. doi: 10.1124/dmd.111.043703. Epub 2012 Jan 19.
Drug Metab Dispos. 2012.
PMID: 22266779
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