Conejo-Garcia A - Search Results

1

Structural basis for binding of cyclic 2-oxoglutarate analogues to factor-inhibiting hypoxia-inducible factor.

Conejo-Garcia A, McDonough MA, Loenarz C, McNeill LA, Hewitson KS, Ge W, Liénard BM, Schofield CJ, Clifton IJ. Conejo-Garcia A, et al. Bioorg Med Chem Lett. 2010 Oct 15;20(20):6125-8. doi: 10.1016/j.bmcl.2010.08.032. Epub 2010 Aug 10. Bioorg Med Chem Lett. 2010. PMID: 20822901

2

A prodrug system for hydroxylamines based on esterase catalysis.

Conejo-Garcia A, Schofield CJ. Conejo-Garcia A, et al. Bioorg Med Chem Lett. 2005 Sep 15;15(18):4004-9. doi: 10.1016/j.bmcl.2005.06.026. Bioorg Med Chem Lett. 2005. PMID: 15990293

3

The inhibition of factor inhibiting hypoxia-inducible factor (FIH) by beta-oxocarboxylic acids.

Banerji B, Conejo-Garcia A, McNeill LA, McDonough MA, Buck MR, Hewitson KS, Oldham NJ, Schofield CJ. Banerji B, et al. Chem Commun (Camb). 2005 Nov 21;(43):5438-40. doi: 10.1039/b510707e. Epub 2005 Oct 4. Chem Commun (Camb). 2005. PMID: 16261239

4

Evaluation of aspirin metabolites as inhibitors of hypoxia-inducible factor hydroxylases.

Lienard BM, Conejo-García A, Stolze I, Loenarz C, Oldham NJ, Ratcliffe PJ, Schofield CJ. Lienard BM, et al. Chem Commun (Camb). 2008 Dec 21;(47):6393-5. doi: 10.1039/b814440k. Epub 2008 Nov 5. Chem Commun (Camb). 2008. PMID: 19048166

5

Selective small molecule probes for the hypoxia inducible factor (HIF) prolyl hydroxylases.

Chowdhury R, Candela-Lena JI, Chan MC, Greenald DJ, Yeoh KK, Tian YM, McDonough MA, Tumber A, Rose NR, Conejo-Garcia A, Demetriades M, Mathavan S, Kawamura A, Lee MK, van Eeden F, Pugh CW, Ratcliffe PJ, Schofield CJ. Chowdhury R, et al. ACS Chem Biol. 2013 Jul 19;8(7):1488-96. doi: 10.1021/cb400088q. Epub 2013 Jun 12. ACS Chem Biol. 2013. PMID: 23683440

6

N-aryltetrahydroisoquinoline derivatives as HA-CD44 interaction inhibitors: Design, synthesis, computational studies, and antitumor effect.

Espejo-Román JM, Rubio-Ruiz B, Chayah-Ghaddab M, Vega-Gutierrez C, García-García G, Muguruza-Montero A, Domene C, Sánchez-Martín RM, Cruz-López O, Conejo-García A. Espejo-Román JM, et al. Among authors: conejo garcia a. Eur J Med Chem. 2023 Oct 5;258:115570. doi: 10.1016/j.ejmech.2023.115570. Epub 2023 Jun 26. Eur J Med Chem. 2023. PMID: 37413883 Free article.

7

Plasmodium falciparum Choline Kinase Inhibition Leads to a Major Decrease in Phosphatidylethanolamine Causing Parasite Death.

Serrán-Aguilera L, Denton H, Rubio-Ruiz B, López-Gutiérrez B, Entrena A, Izquierdo L, Smith TK, Conejo-García A, Hurtado-Guerrero R. Serrán-Aguilera L, et al. Sci Rep. 2016 Sep 12;6:33189. doi: 10.1038/srep33189. Sci Rep. 2016. PMID: 27616047 Free PMC article.

8

Recent advances in the design of choline kinase α inhibitors and the molecular basis of their inhibition.

Rubio-Ruiz B, Serrán-Aguilera L, Hurtado-Guerrero R, Conejo-García A. Rubio-Ruiz B, et al. Among authors: conejo garcia a. Med Res Rev. 2021 Mar;41(2):902-927. doi: 10.1002/med.21746. Epub 2020 Oct 25. Med Res Rev. 2021. PMID: 33103259 Free article. Review.

9

Discovery of a new binding site on human choline kinase α1: design, synthesis, crystallographic studies, and biological evaluation of asymmetrical bispyridinium derivatives.

Rubio-Ruiz B, Figuerola-Conchas A, Ramos-Torrecillas J, Capitán-Cañadas F, Ríos-Marco P, Carrasco MP, Gallo MÁ, Espinosa A, Marco C, Ruiz C, Entrena A, Hurtado-Guerrero R, Conejo-García A. Rubio-Ruiz B, et al. J Med Chem. 2014 Jan 23;57(2):507-15. doi: 10.1021/jm401665x. Epub 2014 Jan 14. J Med Chem. 2014. PMID: 24387243

10

Conformational dynamics of a bispyridinium cyclophane.

Conejo-García A, Campos JM, Entrena A, Sánchez-Martín RM, Gallo MA, Espinosa A. Conejo-García A, et al. J Org Chem. 2003 Oct 31;68(22):8697-9. doi: 10.1021/jo0301292. J Org Chem. 2003. PMID: 14575504

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