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Dipeptidyl peptidase-4 inhibitors administered in combination with metformin result in an additive increase in the plasma concentration of active GLP-1.
Clin Pharmacol Ther. 2010 Dec;88(6):801-8. doi: 10.1038/clpt.2010.184. Epub 2010 Nov 3.
Clin Pharmacol Ther. 2010.
PMID: 21048706
Clinical Trial.
A comparative study of the binding properties, dipeptidyl peptidase-4 (DPP-4) inhibitory activity and glucose-lowering efficacy of the DPP-4 inhibitors alogliptin, linagliptin, saxagliptin, sitagliptin and vildagliptin in mice.
Berger JP, SinhaRoy R, Pocai A, Kelly TM, Scapin G, Gao YD, Pryor KAD, Wu JK, Eiermann GJ, Xu SS, Zhang X, Tatosian DA, Weber AE, Thornberry NA, Carr RD.
Berger JP, et al. Among authors: pryor kad.
Endocrinol Diabetes Metab. 2017 Nov 24;1(1):e00002. doi: 10.1002/edm2.2. eCollection 2018 Jan.
Endocrinol Diabetes Metab. 2017.
PMID: 30815539
Free PMC article.
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Crystallization and preliminary X-ray analysis of the Escherichia coli UDP-MurNAc-tripeptide D-alanyl-D-alanine-adding enzyme (MurF).
Yan Y, Munshi S, Li Y, Pryor KA, Marsilio F, Leiting B.
Yan Y, et al. Among authors: pryor ka.
Acta Crystallogr D Biol Crystallogr. 1999 Dec;55(Pt 12):2033-4. doi: 10.1107/s0907444999011786.
Acta Crystallogr D Biol Crystallogr. 1999.
PMID: 10666581
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Dipeptidyl peptidase IV inhibition for the treatment of type 2 diabetes: potential importance of selectivity over dipeptidyl peptidases 8 and 9.
Lankas GR, Leiting B, Roy RS, Eiermann GJ, Beconi MG, Biftu T, Chan CC, Edmondson S, Feeney WP, He H, Ippolito DE, Kim D, Lyons KA, Ok HO, Patel RA, Petrov AN, Pryor KA, Qian X, Reigle L, Woods A, Wu JK, Zaller D, Zhang X, Zhu L, Weber AE, Thornberry NA.
Lankas GR, et al. Among authors: pryor ka.
Diabetes. 2005 Oct;54(10):2988-94. doi: 10.2337/diabetes.54.10.2988.
Diabetes. 2005.
PMID: 16186403
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