Angelaud R - Search Results

1

A practical synthesis of renin inhibitor MK-1597 (ACT-178882) via catalytic enantioselective hydrogenation and epimerization of piperidine intermediate.

Molinaro C, Shultz S, Roy A, Lau S, Trinh T, Angelaud R, O'Shea PD, Abele S, Cameron M, Corley E, Funel JA, Steinhuebel D, Weisel M, Krska S. Molinaro C, et al. Among authors: angelaud r. J Org Chem. 2011 Feb 18;76(4):1062-71. doi: 10.1021/jo102070e. Epub 2011 Jan 20. J Org Chem. 2011. PMID: 21250716

2

Synthesis of a beta-amino acid pharmacophore via a beta-lactam intermediate.

Angelaud R, Zhong YL, Maligres P, Lee J, Askin D. Angelaud R, et al. J Org Chem. 2005 Mar 4;70(5):1949-52. doi: 10.1021/jo048249c. J Org Chem. 2005. PMID: 15730331

3

A practical synthesis of alpha-aryl methyl ketones via a transition-metal-free Meerwein arylation.

Molinaro C, Mowat J, Gosselin F, O'Shea PD, Marcoux JF, Angelaud R, Davies IW. Molinaro C, et al. Among authors: angelaud r. J Org Chem. 2007 Mar 2;72(5):1856-8. doi: 10.1021/jo062483g. Epub 2007 Jan 31. J Org Chem. 2007. PMID: 17263583

4

Remote electronic control in the regioselective reduction of succinimides: a practical, scalable synthesis of Ep4 antagonist MF-310.

Molinaro C, Gauvreau D, Hughes G, Lau S, Lauzon S, Angelaud R, O'Shea PD, Janey J, Palucki M, Hoerrner SR, Raab CE, Sidler RR, Belley M, Han Y. Molinaro C, et al. Among authors: angelaud r. J Org Chem. 2009 Sep 4;74(17):6863-6. doi: 10.1021/jo901267x. J Org Chem. 2009. PMID: 19663395

5

Preparative scale synthesis of the biaryl core of anacetrapib via a ruthenium-catalyzed direct arylation reaction: unexpected effect of solvent impurity on the arylation reaction.

Ouellet SG, Roy A, Molinaro C, Angelaud R, Marcoux JF, O'Shea PD, Davies IW. Ouellet SG, et al. Among authors: angelaud r. J Org Chem. 2011 Mar 4;76(5):1436-9. doi: 10.1021/jo1018574. Epub 2011 Feb 1. J Org Chem. 2011. PMID: 21284400

6

Stereoselective Synthesis of the IDO Inhibitor Navoximod.

St-Jean F, Angelaud R, Bachmann S, Carrera DE, Remarchuk T, Piechowicz KA, Niedermann K, Iding H, Meier R, Hou H, Sirois LE, Xu J, Olbrich M, Rege P, Guillemot-Plass M, Gosselin F. St-Jean F, et al. Among authors: angelaud r. J Org Chem. 2022 Apr 1;87(7):4955-4960. doi: 10.1021/acs.joc.1c02994. Epub 2022 Mar 23. J Org Chem. 2022. PMID: 35317556

7

Magnesium Ethoxide Promoted Conversion of Nitriles to Amidines and Its Application in 5,6-Dihydroimidazobenzoxazepine Synthesis.

Dalziel ME, Deichert JA, Carrera DE, Beaudry D, Han C, Zhang H, Angelaud R. Dalziel ME, et al. Among authors: angelaud r. Org Lett. 2018 May 4;20(9):2624-2627. doi: 10.1021/acs.orglett.8b00824. Epub 2018 Apr 24. Org Lett. 2018. PMID: 29687714

8

Serendipitous discovery of a pH-dependant atropisomer bond rotation: toward a write-protectable chiral molecular switch?

Welch CJ, Biba M, Pye P, Angelaud R, Egbertson M. Welch CJ, et al. Among authors: angelaud r. J Chromatogr B Analyt Technol Biomed Life Sci. 2008 Nov 1;875(1):118-21. doi: 10.1016/j.jchromb.2008.08.028. J Chromatogr B Analyt Technol Biomed Life Sci. 2008. PMID: 18819851

9

Second-Generation Atroposelective Synthesis of KRAS G12C Covalent Inhibitor GDC-6036.

Xu J, Lim NK, Timmerman JC, Shen J, Clagg K, Orcel U, Bigler R, Trachsel E, Meier R, White NA, Burkhard JA, Sirois LE, Tian Q, Angelaud R, Bachmann S, Zhang H, Gosselin F. Xu J, et al. Among authors: angelaud r. Org Lett. 2023 May 19;25(19):3417-3422. doi: 10.1021/acs.orglett.3c00961. Epub 2023 May 10. Org Lett. 2023. PMID: 37162129

10

Asymmetric activation of chiral alkoxyzinc catalysts by chiral nitrogen activators for dialkylzinc addition to aldehydes: super high-throughput screening of combinatorial libraries of chiral ligands and activators by HPLC-CD/UV and HPLC-OR/RIU systems.

Mikami K, Angelaud R, Ding K, Ishii A, Tanaka A, Sawada N, Kudo K, Senda M. Mikami K, et al. Among authors: angelaud r. Chemistry. 2001 Feb 2;7(3):730-7. doi: 10.1002/1521-3765(20010202)7:3<730::aid-chem730>3.0.co;2-1. Chemistry. 2001. PMID: 11261671

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