Search Page
Save citations to file
Email citations
Send citations to clipboard
Add to Collections
Add to My Bibliography
Create a file for external citation management software
Your saved search
Your RSS Feed
Search Results
8 results
Filters applied: . Clear all
Results are displayed in a computed author sort order.
The Results By Year timeline is not available.
Page 1
Screening and identification of a novel class of TGF-β type 1 receptor kinase inhibitor.
J Biomol Screen. 2011 Aug;16(7):724-33. doi: 10.1177/1087057111405846. Epub 2011 Apr 26.
J Biomol Screen. 2011.
PMID: 21521800
ASK1 contributes to fibrosis and dysfunction in models of kidney disease.
Liles JT, Corkey BK, Notte GT, Budas GR, Lansdon EB, Hinojosa-Kirschenbaum F, Badal SS, Lee M, Schultz BE, Wise S, Pendem S, Graupe M, Castonguay L, Koch KA, Wong MH, Papalia GA, French DM, Sullivan T, Huntzicker EG, Ma FY, Nikolic-Paterson DJ, Altuhaifi T, Yang H, Fogo AB, Breckenridge DG.
Liles JT, et al.
J Clin Invest. 2018 Oct 1;128(10):4485-4500. doi: 10.1172/JCI99768. Epub 2018 Jul 19.
J Clin Invest. 2018.
PMID: 30024858
Free PMC article.
Item in Clipboard
Conformational analysis and receptor docking of N-[(1S,2S)-3-(4-chlorophenyl)-2-(3-cyanophenyl)-1-methylpropyl]-2-methyl-2-{[5-(trifluoromethyl)pyridin-2-yl]oxy}propanamide (taranabant, MK-0364), a novel, acyclic cannabinoid-1 receptor inverse agonist.
Lin LS, Ha S, Ball RG, Tsou NN, Castonguay LA, Doss GA, Fong TM, Shen CP, Xiao JC, Goulet MT, Hagmann WK.
Lin LS, et al. Among authors: castonguay la.
J Med Chem. 2008 Apr 10;51(7):2108-14. doi: 10.1021/jm7014974. Epub 2008 Mar 12.
J Med Chem. 2008.
PMID: 18333607
Item in Clipboard
Bioisosteric replacement of anilide with benzoxazole: potent and orally bioavailable antagonists of VLA-4.
Lin LS, Lanza TJ Jr, Castonguay LA, Kamenecka T, McCauley E, Van Riper G, Egger LA, Mumford RA, Tong X, MacCoss M, Schmidt JA, Hagmann WK.
Lin LS, et al. Among authors: castonguay la.
Bioorg Med Chem Lett. 2004 May 3;14(9):2331-4. doi: 10.1016/j.bmcl.2004.01.098.
Bioorg Med Chem Lett. 2004.
PMID: 15081035
Item in Clipboard
Binding of 2-aryl-4-(piperidin-1-yl)butanamines and 1,3,4-trisubstituted pyrrolidines to human CCR5: a molecular modeling-guided mutagenesis study of the binding pocket.
Castonguay LA, Weng Y, Adolfsen W, Di Salvo J, Kilburn R, Caldwell CG, Daugherty BL, Finke PE, Hale JJ, Lynch CL, Mills SG, MacCoss M, Springer MS, DeMartino JA.
Castonguay LA, et al.
Biochemistry. 2003 Feb 18;42(6):1544-50. doi: 10.1021/bi026639s.
Biochemistry. 2003.
PMID: 12578367
Item in Clipboard
Prediction of q-values and conformations of gadolinium chelates for magnetic resonance imaging.
Castonguay LA, Treasurywala AM, Caulfield TJ, Jaeger EP, Kellar KE.
Castonguay LA, et al.
Bioconjug Chem. 1999 Nov-Dec;10(6):958-64. doi: 10.1021/bc990027b.
Bioconjug Chem. 1999.
PMID: 10563764
Item in Clipboard
Novel inhibitors of potassium ion channels on human T lymphocytes.
Michne WF, Guiles JW, Treasurywala AM, Castonguay LA, Weigelt CA, Oconnor B, Volberg WA, Grant AM, Chadwick CC, Krafte DS, et al.
Michne WF, et al. Among authors: castonguay la.
J Med Chem. 1995 May 26;38(11):1877-83. doi: 10.1021/jm00011a007.
J Med Chem. 1995.
PMID: 7540207
Item in Clipboard
A proposed structural model of domain 1 of fasciclin III neural cell adhesion protein based on an inverse folding algorithm.
Castonguay LA, Bryant SH, Snow PM, Fetrow JS.
Castonguay LA, et al.
Protein Sci. 1995 Mar;4(3):472-83. doi: 10.1002/pro.5560040314.
Protein Sci. 1995.
PMID: 7795530
Free PMC article.
Item in Clipboard
Cite
Cite