Velaparthi S - Search Results

1

Discovery, synthesis and SAR analysis of novel selective small molecule S1P4-R agonists based on a (2Z,5Z)-5-((pyrrol-3-yl)methylene)-3-alkyl-2-(alkylimino)thiazolidin-4-one chemotype.

Urbano M, Guerrero M, Velaparthi S, Crisp M, Chase P, Hodder P, Schaeffer MT, Brown S, Rosen H, Roberts E. Urbano M, et al. Among authors: velaparthi s. Bioorg Med Chem Lett. 2011 Nov 15;21(22):6739-45. doi: 10.1016/j.bmcl.2011.09.049. Epub 2011 Sep 20. Bioorg Med Chem Lett. 2011. PMID: 21982495 Free PMC article.

2

Discovery, design and synthesis of the first reported potent and selective sphingosine-1-phosphate 4 (S1P4) receptor antagonists.

Guerrero M, Urbano M, Velaparthi S, Zhao J, Schaeffer MT, Brown S, Rosen H, Roberts E. Guerrero M, et al. Among authors: velaparthi s. Bioorg Med Chem Lett. 2011 Jun 15;21(12):3632-6. doi: 10.1016/j.bmcl.2011.04.097. Epub 2011 Apr 28. Bioorg Med Chem Lett. 2011. PMID: 21570287 Free PMC article.

3

SAR analysis of innovative selective small molecule antagonists of sphingosine-1-phosphate 4 (S1P₄) receptor.

Urbano M, Guerrero M, Zhao J, Velaparthi S, Schaeffer MT, Brown S, Rosen H, Roberts E. Urbano M, et al. Among authors: velaparthi s. Bioorg Med Chem Lett. 2011 Sep 15;21(18):5470-4. doi: 10.1016/j.bmcl.2011.06.132. Epub 2011 Jul 13. Bioorg Med Chem Lett. 2011. PMID: 21783362 Free PMC article.

4

Design, synthesis and SAR analysis of novel potent and selective small molecule antagonists of NPBWR1 (GPR7).

Urbano M, Guerrero M, Zhao J, Velaparthi S, Saldanha SA, Chase P, Wang Z, Civelli O, Hodder P, Schaeffer MT, Brown S, Rosen H, Roberts E. Urbano M, et al. Among authors: velaparthi s. Bioorg Med Chem Lett. 2012 Dec 1;22(23):7135-41. doi: 10.1016/j.bmcl.2012.09.074. Epub 2012 Oct 2. Bioorg Med Chem Lett. 2012. PMID: 23079522 Free PMC article.

5

Design, synthesis, docking, and biological evaluation of novel diazide-containing isoxazole- and pyrazole-based histone deacetylase probes.

Neelarapu R, Holzle DL, Velaparthi S, Bai H, Brunsteiner M, Blond SY, Petukhov PA. Neelarapu R, et al. Among authors: velaparthi s. J Med Chem. 2011 Jul 14;54(13):4350-64. doi: 10.1021/jm2001025. Epub 2011 Jun 2. J Med Chem. 2011. PMID: 21548582 Free PMC article.

6

5-tert-butyl-N-pyrazol-4-yl-4,5,6,7-tetrahydrobenzo[d]isoxazole-3-carboxamide derivatives as novel potent inhibitors of Mycobacterium tuberculosis pantothenate synthetase: initiating a quest for new antitubercular drugs.

Velaparthi S, Brunsteiner M, Uddin R, Wan B, Franzblau SG, Petukhov PA. Velaparthi S, et al. J Med Chem. 2008 Apr 10;51(7):1999-2002. doi: 10.1021/jm701372r. Epub 2008 Mar 13. J Med Chem. 2008. PMID: 18335974 Review.

7

Binding ensemble profiling with photoaffinity labeling (BEProFL) approach: mapping the binding poses of HDAC8 inhibitors.

He B, Velaparthi S, Pieffet G, Pennington C, Mahesh A, Holzle DL, Brunsteiner M, van Breemen R, Blond SY, Petukhov PA. He B, et al. Among authors: velaparthi s. J Med Chem. 2009 Nov 26;52(22):7003-13. doi: 10.1021/jm9005077. J Med Chem. 2009. PMID: 19886628 Free PMC article.

8

Arylation of rhodium(II) azavinyl carbenes with boronic acids.

Selander N, Worrell BT, Chuprakov S, Velaparthi S, Fokin VV. Selander N, et al. Among authors: velaparthi s. J Am Chem Soc. 2012 Sep 12;134(36):14670-3. doi: 10.1021/ja3062453. Epub 2012 Aug 28. J Am Chem Soc. 2012. PMID: 22913576 Free PMC article.

9

Chirality and template-mediated induction of helical preferences in achiral β-peptides.

Sharma GV, Kodeti SR, Dutta SK, Velaparthi S, Narsimulu K, Anjaiah G, Jeelani Basha S, Kunwar AC. Sharma GV, et al. Among authors: velaparthi s. Chemistry. 2012 Dec 7;18(50):16046-60. doi: 10.1002/chem.201201892. Epub 2012 Oct 30. Chemistry. 2012. PMID: 23111903

10

Probe Development Efforts to Identify Novel Agonists of the Sphingosine 1-phosphate Receptor 4 (S1P4).

Guerrero M, Urbano M, Velaparthi S, Zhao J, Schaeffer MT, Brown SJ, Crisp M, Ferguson J, Roberts E, Oldstone M, Hodder P, Rosen H. Guerrero M, et al. Among authors: velaparthi s. 2010 Oct 12 [updated 2011 Dec 12]. In: Probe Reports from the NIH Molecular Libraries Program [Internet]. Bethesda (MD): National Center for Biotechnology Information (US); 2010–. 2010 Oct 12 [updated 2011 Dec 12]. In: Probe Reports from the NIH Molecular Libraries Program [Internet]. Bethesda (MD): National Center for Biotechnology Information (US); 2010–. PMID: 22834032 Free Books & Documents. Review.

Save citations to file

Email citations

Send citations to clipboard

Add to Collections

Add to My Bibliography

Create a file for external citation management software

Your saved search

Your RSS Feed

My NCBI Filters

Text availability

Article attribute

Article type

Publication date

14 results

Search Page