Dack K - Search Results

1

Use of libraries to access new chemical space: applications to CRTH2.

Abid Masood M, Gardner M, Dack K, Winpenny D, Lunn G. Abid Masood M, et al. Among authors: dack k. Bioorg Med Chem Lett. 2012 Jun 1;22(11):3682-7. doi: 10.1016/j.bmcl.2012.04.041. Epub 2012 Apr 20. Bioorg Med Chem Lett. 2012. PMID: 22560471

2

Optimisation of a pyrazole series of progesterone antagonists; Part 1.

Dack KN, Skerratt S, Johnson PS, Bradley PA, Marsh IR. Dack KN, et al. Bioorg Med Chem Lett. 2010 Jun 1;20(11):3384-6. doi: 10.1016/j.bmcl.2010.04.018. Epub 2010 Apr 13. Bioorg Med Chem Lett. 2010. PMID: 20430618

3

The design and synthesis of a novel series of indole derived selective ET(A) antagonists.

Rawson DJ, Dack KN, Dickinson RP, James K. Rawson DJ, et al. Among authors: dack kn. Bioorg Med Chem Lett. 2002 Jan 21;12(2):125-8. doi: 10.1016/s0960-894x(01)00660-6. Bioorg Med Chem Lett. 2002. PMID: 11755336

4

A novel series of highly selective inhibitors of MMP-3.

Whitlock GA, Dack KN, Dickinson RP, Lewis ML. Whitlock GA, et al. Bioorg Med Chem Lett. 2007 Dec 15;17(24):6750-3. doi: 10.1016/j.bmcl.2007.10.042. Epub 2007 Oct 17. Bioorg Med Chem Lett. 2007. PMID: 18029177

5

Discovery of PF-184563, a potent and selective V1a antagonist for the treatment of dysmenorrhoea. The influence of compound flexibility on microsomal stability.

Johnson PS, Ryckmans T, Bryans J, Beal DM, Dack KN, Feeder N, Harrison A, Lewis M, Mason HJ, Mills J, Newman J, Pasquinet C, Rawson DJ, Roberts LR, Russell R, Spark D, Stobie A, Underwood TJ, Ward R, Wheeler S. Johnson PS, et al. Bioorg Med Chem Lett. 2011 Oct 1;21(19):5684-7. doi: 10.1016/j.bmcl.2011.08.038. Epub 2011 Aug 12. Bioorg Med Chem Lett. 2011. PMID: 21885275

6

Synthesis and evaluation of heteroarylalanine diacids as potent and selective neutral endopeptidase inhibitors.

Glossop MS, Bazin RJ, Dack KN, Fox DN, MacDonald GA, Mills M, Owen DR, Phillips C, Reeves KA, Ringer TJ, Strang RS, Watson CA. Glossop MS, et al. Bioorg Med Chem Lett. 2011 Jun 1;21(11):3404-6. doi: 10.1016/j.bmcl.2011.03.109. Epub 2011 Apr 5. Bioorg Med Chem Lett. 2011. PMID: 21515054

7

Acidic triazoles as soluble guanylate cyclase stimulators.

Roberts LR, Bradley PA, Bunnage ME, England KS, Fairman D, Fobian YM, Fox DN, Gymer GE, Heasley SE, Molette J, Smith GL, Schmidt MA, Tones MA, Dack KN. Roberts LR, et al. Bioorg Med Chem Lett. 2011 Nov 1;21(21):6515-8. doi: 10.1016/j.bmcl.2011.08.071. Epub 2011 Aug 28. Bioorg Med Chem Lett. 2011. PMID: 21924901

8

Thromboxane modulating agents. 4. Design and synthesis of 3-(2-[[(4-chlorophenyl)sulfonyl]-amino]ethyl)benzenepropanoic acid derivatives as potent thromboxane receptor antagonists.

Dack KN, Dickinson RP, Long CJ, Steele J. Dack KN, et al. Bioorg Med Chem Lett. 1998 Aug 18;8(16):2061-6. doi: 10.1016/s0960-894x(98)00242-x. Bioorg Med Chem Lett. 1998. PMID: 9873486

9

Discovery of aryloxy tetramethylcyclobutanes as novel androgen receptor antagonists.

Guo C, Linton A, Kephart S, Ornelas M, Pairish M, Gonzalez J, Greasley S, Nagata A, Burke BJ, Edwards M, Hosea N, Kang P, Hu W, Engebretsen J, Briere D, Shi M, Gukasyan H, Richardson P, Dack K, Underwood T, Johnson P, Morell A, Felstead R, Kuruma H, Matsimoto H, Zoubeidi A, Gleave M, Los G, Fanjul AN. Guo C, et al. Among authors: dack k. J Med Chem. 2011 Nov 10;54(21):7693-704. doi: 10.1021/jm201059s. Epub 2011 Oct 7. J Med Chem. 2011. PMID: 21936524

10

Thromboxane modulating agents. 3. 1H-imidazol-1-ylalkyl- and 3-pyridinylalkyl-substituted 3-[2-[(arylsulfonyl)amino]ethyl]benzenepropanoic acid derivatives as dual thromboxane synthase inhibitor/thromboxane receptor antagonists.

Dickinson RP, Dack KN, Long CJ, Steele J. Dickinson RP, et al. Among authors: dack kn. J Med Chem. 1997 Oct 10;40(21):3442-52. doi: 10.1021/jm9702793. J Med Chem. 1997. PMID: 9341919

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