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The optimization of pyridazinone series of glucan synthase inhibitors.
Bioorg Med Chem Lett. 2012 Aug 15;22(16):5268-71. doi: 10.1016/j.bmcl.2012.06.091. Epub 2012 Jul 4.
Bioorg Med Chem Lett. 2012.
PMID: 22818082
Bioavailable pyrrolo-benzo-1,4-diazines as Na(v)1.7 sodium channel blockers for the treatment of pain.
Yang SW, Ho GD, Tulshian D, Bercovici A, Tan Z, Hanisak J, Brumfield S, Matasi J, Sun X, Sakwa SA, Herr RJ, Zhou X, Bridal T, Urban M, Vivian J, Rindgen D, Sorota S.
Yang SW, et al. Among authors: sakwa sa.
Bioorg Med Chem Lett. 2014 Nov 1;24(21):4958-62. doi: 10.1016/j.bmcl.2014.09.038. Epub 2014 Sep 19.
Bioorg Med Chem Lett. 2014.
PMID: 25288187
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Iminopyrimidinones: a novel pharmacophore for the development of orally active renin inhibitors.
McKittrick BA, Caldwell JP, Bara T, Boykow G, Chintala M, Clader J, Czarniecki M, Courneya B, Duffy R, Fleming L, Giessert R, Greenlee WJ, Heap C, Hong L, Huang Y, Iserloh U, Josien H, Khan T, Korfmacher W, Liang X, Mazzola R, Mitra S, Moore K, Orth P, Rajagopalan M, Roy S, Sakwa S, Strickland C, Vaccaro H, Voigt J, Wang H, Wong J, Zhang R, Zych A.
McKittrick BA, et al.
Bioorg Med Chem Lett. 2015 Apr 1;25(7):1592-6. doi: 10.1016/j.bmcl.2015.02.003. Epub 2015 Feb 10.
Bioorg Med Chem Lett. 2015.
PMID: 25728416
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Design and synthesis of aminothiazole modulators of the gamma-secretase enzyme.
Rynearson KD, Buckle RN, Barnes KD, Herr RJ, Mayhew NJ, Paquette WD, Sakwa SA, Nguyen PD, Johnson G, Tanzi RE, Wagner SL.
Rynearson KD, et al. Among authors: sakwa sa.
Bioorg Med Chem Lett. 2016 Aug 15;26(16):3928-37. doi: 10.1016/j.bmcl.2016.07.011. Epub 2016 Jul 6.
Bioorg Med Chem Lett. 2016.
PMID: 27426299
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Design and synthesis of novel methoxypyridine-derived gamma-secretase modulators.
Rynearson KD, Buckle RN, Herr RJ, Mayhew NJ, Chen X, Paquette WD, Sakwa SA, Yang J, Barnes KD, Nguyen P, Mobley WC, Johnson G, Lin JH, Tanzi RE, Wagner SL.
Rynearson KD, et al. Among authors: sakwa sa.
Bioorg Med Chem. 2020 Nov 15;28(22):115734. doi: 10.1016/j.bmc.2020.115734. Epub 2020 Sep 1.
Bioorg Med Chem. 2020.
PMID: 33007551
Free PMC article.
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Synthesis and Biological Evaluation of N-((1-(4-(Sulfonyl)piperazin-1-yl)cycloalkyl)methyl)benzamide Inhibitors of Glycine Transporter-1.
Cioffi CL, Liu S, Wolf MA, Guzzo PR, Sadalapure K, Parthasarathy V, Loong DT, Maeng JH, Carulli E, Fang X, Karunakaran K, Matta L, Choo SH, Panduga S, Buckle RN, Davis RN, Sakwa SA, Gupta P, Sargent BJ, Moore NA, Luche MM, Carr GJ, Khmelnitsky YL, Ismail J, Chung M, Bai M, Leong WY, Sachdev N, Swaminathan S, Mhyre AJ.
Cioffi CL, et al. Among authors: sakwa sa.
J Med Chem. 2016 Sep 22;59(18):8473-94. doi: 10.1021/acs.jmedchem.6b00914. Epub 2016 Sep 9.
J Med Chem. 2016.
PMID: 27559615
Free article.
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A concise palladium-catalyzed carboamination route to (+/-)-tylophorine.
Rossiter LM, Slater ML, Giessert RE, Sakwa SA, Herr RJ.
Rossiter LM, et al. Among authors: sakwa sa.
J Org Chem. 2009 Dec 18;74(24):9554-7. doi: 10.1021/jo902114u.
J Org Chem. 2009.
PMID: 19919084
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