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The optimization of pyridazinone series of glucan synthase inhibitors.
Bioorg Med Chem Lett. 2012 Aug 15;22(16):5268-71. doi: 10.1016/j.bmcl.2012.06.091. Epub 2012 Jul 4.
Bioorg Med Chem Lett. 2012.
PMID: 22818082
SAR studies of pyridazinone derivatives as novel glucan synthase inhibitors.
Zhou G, Ting PC, Aslanian R, Cao J, Kim DW, Kuang R, Lee JF, Schwerdt J, Wu H, Herr RJ, Zych AJ, Yang J, Lam S, Wainhaus S, Black TA, McNicholas PM, Xu Y, Walker SS.
Zhou G, et al. Among authors: zych aj.
Bioorg Med Chem Lett. 2011 May 15;21(10):2890-3. doi: 10.1016/j.bmcl.2011.03.083. Epub 2011 Mar 30.
Bioorg Med Chem Lett. 2011.
PMID: 21489787
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Lead optimization of a sulfonylurea-based piperazine pyridazinone series of glucan synthase inhibitors.
Zych AJ, Lam SQ, Jenkins DM, Herr RJ, Ting PC, Lee JF, Kuang R, Wu H, Kim DW, Aslanian RG, Wainhaus S, Black TA, Cacciapuoti A, McNicholas PM, Xu Y, Walker SS.
Zych AJ, et al.
Bioorg Med Chem Lett. 2012 Jul 15;22(14):4896-9. doi: 10.1016/j.bmcl.2012.04.127. Epub 2012 May 17.
Bioorg Med Chem Lett. 2012.
PMID: 22687744
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Iminopyrimidinones: a novel pharmacophore for the development of orally active renin inhibitors.
McKittrick BA, Caldwell JP, Bara T, Boykow G, Chintala M, Clader J, Czarniecki M, Courneya B, Duffy R, Fleming L, Giessert R, Greenlee WJ, Heap C, Hong L, Huang Y, Iserloh U, Josien H, Khan T, Korfmacher W, Liang X, Mazzola R, Mitra S, Moore K, Orth P, Rajagopalan M, Roy S, Sakwa S, Strickland C, Vaccaro H, Voigt J, Wang H, Wong J, Zhang R, Zych A.
McKittrick BA, et al.
Bioorg Med Chem Lett. 2015 Apr 1;25(7):1592-6. doi: 10.1016/j.bmcl.2015.02.003. Epub 2015 Feb 10.
Bioorg Med Chem Lett. 2015.
PMID: 25728416
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Assessing the impact of expert knowledge on ICH M7 (Q)SAR predictions. Is expert review still needed?
Jayasekara PS, Skanchy SK, Kim MT, Kumaran G, Mugabe BE, Woodard LE, Yang J, Zych AJ, Kruhlak NL.
Jayasekara PS, et al. Among authors: zych aj.
Regul Toxicol Pharmacol. 2021 Oct;125:105006. doi: 10.1016/j.yrtph.2021.105006. Epub 2021 Jul 14.
Regul Toxicol Pharmacol. 2021.
PMID: 34273441
Free article.
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