Richters A - Search Results

1

Identification of type II and III DDR2 inhibitors.

Richters A, Nguyen HD, Phan T, Simard JR, Grütter C, Engel J, Rauh D. Richters A, et al. J Med Chem. 2014 May 22;57(10):4252-62. doi: 10.1021/jm500167q. Epub 2014 May 5. J Med Chem. 2014. PMID: 24754677

2

Targeting gain of function and resistance mutations in Abl and KIT by hybrid compound design.

Richters A, Ketzer J, Getlik M, Grütter C, Schneider R, Heuckmann JM, Heynck S, Sos ML, Gupta A, Unger A, Schultz-Fademrecht C, Thomas RK, Bauer S, Rauh D. Richters A, et al. J Med Chem. 2013 Jul 25;56(14):5757-72. doi: 10.1021/jm4004076. Epub 2013 Jul 10. J Med Chem. 2013. PMID: 23773153

3

Identification and further development of potent TBK1 inhibitors.

Richters A, Basu D, Engel J, Ercanoglu MS, Balke-Want H, Tesch R, Thomas RK, Rauh D. Richters A, et al. ACS Chem Biol. 2015 Jan 16;10(1):289-98. doi: 10.1021/cb500908d. ACS Chem Biol. 2015. PMID: 25540906

4

Structure-based design and synthesis of covalent-reversible inhibitors to overcome drug resistance in EGFR.

Basu D, Richters A, Rauh D. Basu D, et al. Among authors: richters a. Bioorg Med Chem. 2015 Jun 15;23(12):2767-80. doi: 10.1016/j.bmc.2015.04.038. Epub 2015 Apr 23. Bioorg Med Chem. 2015. PMID: 25975640

5

Targeting Drug Resistance in EGFR with Covalent Inhibitors: A Structure-Based Design Approach.

Engel J, Richters A, Getlik M, Tomassi S, Keul M, Termathe M, Lategahn J, Becker C, Mayer-Wrangowski S, Grütter C, Uhlenbrock N, Krüll J, Schaumann N, Eppmann S, Kibies P, Hoffgaard F, Heil J, Menninger S, Ortiz-Cuaran S, Heuckmann JM, Tinnefeld V, Zahedi RP, Sos ML, Schultz-Fademrecht C, Thomas RK, Kast SM, Rauh D. Engel J, et al. Among authors: richters a. J Med Chem. 2015 Sep 10;58(17):6844-63. doi: 10.1021/acs.jmedchem.5b01082. Epub 2015 Aug 31. J Med Chem. 2015. PMID: 26275028

6

Corrigendum to "Structure-based design and synthesis of covalent-reversible inhibitors to overcome drug resistance in EGFR" [Bioorg. Med. Chem. 23, 2015, 2767-2780].

Basu D, Richters A, Rauh D. Basu D, et al. Among authors: richters a. Bioorg Med Chem. 2015 Aug 1;23(15):5075. doi: 10.1016/j.bmc.2015.06.001. Epub 2015 Jun 10. Bioorg Med Chem. 2015. PMID: 32689707 No abstract available.

7

Proteus in the world of proteins: conformational changes in protein kinases.

Rabiller M, Getlik M, Klüter S, Richters A, Tückmantel S, Simard JR, Rauh D. Rabiller M, et al. Among authors: richters a. Arch Pharm (Weinheim). 2010 Apr;343(4):193-206. doi: 10.1002/ardp.201000028. Arch Pharm (Weinheim). 2010. PMID: 20336692 Review.

8

Targeting GSK3 from Ustilago maydis: type-II kinase inhibitors as potential antifungals.

Grütter C, Simard JR, Mayer-Wrangowski SC, Schreier PH, Pérez-Martín J, Richters A, Getlik M, Gutbrod O, Braun CA, Beck ME, Rauh D. Grütter C, et al. Among authors: richters a. ACS Chem Biol. 2012 Jul 20;7(7):1257-67. doi: 10.1021/cb300128b. Epub 2012 May 15. ACS Chem Biol. 2012. PMID: 22545924

9

Metabolically stable dibenzo[b,e]oxepin-11(6H)-ones as highly selective p38 MAP kinase inhibitors: optimizing anti-cytokine activity in human whole blood.

Baur B, Storch K, Martz KE, Goettert MI, Richters A, Rauh D, Laufer SA. Baur B, et al. Among authors: richters a. J Med Chem. 2013 Nov 14;56(21):8561-78. doi: 10.1021/jm401276h. Epub 2013 Nov 5. J Med Chem. 2013. PMID: 24131218

10

Combining X-ray crystallography and molecular modeling toward the optimization of pyrazolo[3,4-d]pyrimidines as potent c-Src inhibitors active in vivo against neuroblastoma.

Tintori C, Fallacara AL, Radi M, Zamperini C, Dreassi E, Crespan E, Maga G, Schenone S, Musumeci F, Brullo C, Richters A, Gasparrini F, Angelucci A, Festuccia C, Delle Monache S, Rauh D, Botta M. Tintori C, et al. Among authors: richters a. J Med Chem. 2015 Jan 8;58(1):347-61. doi: 10.1021/jm5013159. Epub 2014 Dec 3. J Med Chem. 2015. PMID: 25469771

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