Cheung AW - Search Results

1

Identification of an Adamantyl Azaquinolone JNK Selective Inhibitor.

Haynes NE, Scott NR, Chen LC, Janson CA, Li JK, Lukacs CM, Railkar A, Tozzo E, Whittard T, Brown NF, Cheung AW. Haynes NE, et al. Among authors: cheung aw. ACS Med Chem Lett. 2012 Aug 8;3(9):764-8. doi: 10.1021/ml300175c. eCollection 2012 Sep 13. ACS Med Chem Lett. 2012. PMID: 24900545 Free PMC article.

2

Discovery of orally active carboxylic acid derivatives of 2-phenyl-5-trifluoromethyloxazole-4-carboxamide as potent diacylglycerol acyltransferase-1 inhibitors for the potential treatment of obesity and diabetes.

Qian Y, Wertheimer SJ, Ahmad M, Cheung AW, Firooznia F, Hamilton MM, Hayden S, Li S, Marcopulos N, McDermott L, Tan J, Yun W, Guo L, Pamidimukkala A, Chen Y, Huang KS, Ramsey GB, Whittard T, Conde-Knape K, Taub R, Rondinone CM, Tilley J, Bolin D. Qian Y, et al. Among authors: cheung aw. J Med Chem. 2011 Apr 14;54(7):2433-46. doi: 10.1021/jm101580m. Epub 2011 Mar 17. J Med Chem. 2011. PMID: 21413799

3

Structure-activity relationship of linear peptide Bu-His-DPhe-Arg-Trp-Gly-NH(2) at the human melanocortin-1 and -4 receptors: arginine substitution.

Cheung AW, Danho W, Swistok J, Qi L, Kurylko G, Franco L, Yagaloff K, Chen L. Cheung AW, et al. Bioorg Med Chem Lett. 2002 Sep 2;12(17):2407-10. doi: 10.1016/s0960-894x(02)00459-6. Bioorg Med Chem Lett. 2002. PMID: 12161144

4

Preparation of human Melanocortin-4 receptor agonist libraries: linear peptides X-Y-DPhe7-Arg8-Trp(or 2-Nal)9-Z-NH2.

Cheung AW, Qi L, Gore V, Chu XJ, Bartkovitz D, Kurylko G, Swistok J, Danho W, Chen L, Yagaloff K. Cheung AW, et al. Bioorg Med Chem Lett. 2005 Dec 15;15(24):5504-8. doi: 10.1016/j.bmcl.2005.08.083. Epub 2005 Oct 3. Bioorg Med Chem Lett. 2005. PMID: 16203134

5

Structure-activity relationship of linear peptide Bu-His-DPhe-Arg-Trp-Gly-NH(2) at the human melanocortin-1 and -4 receptors: histidine substitution.

Cheung AW, Danho W, Swistok J, Qi L, Kurylko G, Rowan K, Yeon M, Franco L, Chu XJ, Chen L, Yagaloff K. Cheung AW, et al. Bioorg Med Chem Lett. 2003 Jan 6;13(1):133-7. doi: 10.1016/s0960-894x(02)00830-2. Bioorg Med Chem Lett. 2003. PMID: 12467633

6

Structure-activity relationship of linear peptide Bu-His6-DPhe7-Arg8-Trp9-Gly10-NH2 at the human melanocortin-1 and -4 receptors: DPhe7 and Trp9 substitution.

Danho W, Swistok J, Cheung AW, Kurylko G, Franco L, Chu XJ, Chen L, Yagaloff K. Danho W, et al. Among authors: cheung aw. Bioorg Med Chem Lett. 2003 Feb 24;13(4):649-52. doi: 10.1016/s0960-894x(02)01052-1. Bioorg Med Chem Lett. 2003. PMID: 12639550

7

Discovery of 1-amino-4-phenylcyclohexane-1-carboxylic acid and its influence on agonist selectivity between human melanocortin-4 and -1 receptors in linear pentapeptides.

Chu XJ, Bartkovitz D, Danho W, Swistok J, Cheung AW, Kurylko G, Rowan K, Yeon M, Franco L, Qi L, Chen L, Yagaloff K. Chu XJ, et al. Among authors: cheung aw. Bioorg Med Chem Lett. 2005 Nov 15;15(22):4910-4. doi: 10.1016/j.bmcl.2005.08.012. Bioorg Med Chem Lett. 2005. PMID: 16169218

8

A predictive pharmacophore model of human melanocortin-4 receptor as derived from the solution structures of cyclic peptides.

Sun H, Greeley DN, Chu XJ, Cheung A, Danho W, Swistok J, Wang Y, Zhao C, Chen L, Fry DC. Sun H, et al. Bioorg Med Chem. 2004 May 15;12(10):2671-7. doi: 10.1016/j.bmc.2004.03.017. Bioorg Med Chem. 2004. PMID: 15110848

9

Structure-activity relationship of cyclic peptide penta-c[Asp-His(6)-DPhe(7)-Arg(8)-Trp(9)-Lys]-NH(2) at the human melanocortin-1 and -4 receptors: His(6) substitution.

Cheung AW, Danho W, Swistok J, Qi L, Kurylko G, Rowan K, Yeon M, Franco L, Chu XJ, Chen L, Yagaloff K. Cheung AW, et al. Bioorg Med Chem Lett. 2003 Apr 7;13(7):1307-11. doi: 10.1016/s0960-894x(03)00114-8. Bioorg Med Chem Lett. 2003. PMID: 12657270

10

7-Phenyl-pyrido[2,3-d]pyrimidine-2,4-diamines: novel and highly selective protein tyrosine phosphatase 1B inhibitors.

Cheung AW, Banner B, Bose J, Kim K, Li S, Marcopulos N, Orzechowski L, Sergi JA, Thakkar KC, Wang BB, Yun W, Zwingelstein C, Berthel S, Olivier AR. Cheung AW, et al. Bioorg Med Chem Lett. 2012 Dec 15;22(24):7518-22. doi: 10.1016/j.bmcl.2012.10.035. Epub 2012 Oct 16. Bioorg Med Chem Lett. 2012. PMID: 23122867

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