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Discovery of a Selective TRPM8 Antagonist with Clinical Efficacy in Cold-Related Pain.
ACS Med Chem Lett. 2015 Jan 30;6(4):419-24. doi: 10.1021/ml500479v. eCollection 2015 Apr 9.
ACS Med Chem Lett. 2015.
PMID: 25893043
Free PMC article.
Pyrimido[4,5-d]azepines as potent and selective 5-HT2C receptor agonists: design, synthesis, and evaluation of PF-3246799 as a treatment for urinary incontinence.
Andrews MD, Fish PV, Blagg J, Brabham TK, Brennan PE, Bridgeland A, Brown AD, Bungay PJ, Conlon KM, Edmunds NJ, af Forselles K, Gibbons CP, Green MP, Hanton G, Holbrook M, Jessiman AS, McIntosh K, McMurray G, Nichols CL, Root JA, Storer RI, Sutton MR, Ward RV, Westbrook D, Whitlock GA.
Andrews MD, et al. Among authors: af forselles k.
Bioorg Med Chem Lett. 2011 May 1;21(9):2715-20. doi: 10.1016/j.bmcl.2010.11.120. Epub 2010 Dec 4.
Bioorg Med Chem Lett. 2011.
PMID: 21195614
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In vitro and in vivo characterization of PF-04418948, a novel, potent and selective prostaglandin EP₂ receptor antagonist.
af Forselles KJ, Root J, Clarke T, Davey D, Aughton K, Dack K, Pullen N.
af Forselles KJ, et al.
Br J Pharmacol. 2011 Dec;164(7):1847-56. doi: 10.1111/j.1476-5381.2011.01495.x.
Br J Pharmacol. 2011.
PMID: 21595651
Free PMC article.
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Prostanoid receptors mediating contraction in rat, macaque and human bladder smooth muscle in vitro.
Root JA, Davey DA, Af Forselles KJ.
Root JA, et al. Among authors: af forselles kj.
Eur J Pharmacol. 2015 Dec 15;769:274-9. doi: 10.1016/j.ejphar.2015.11.030. Epub 2015 Nov 25.
Eur J Pharmacol. 2015.
PMID: 26607459
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