Halland N - Search Results

1

G Protein-Coupled Receptor 119 (GPR119) Agonists for the Treatment of Diabetes: Recent Progress and Prevailing Challenges.

Ritter K, Buning C, Halland N, Pöverlein C, Schwink L. Ritter K, et al. Among authors: halland n. J Med Chem. 2016 Apr 28;59(8):3579-92. doi: 10.1021/acs.jmedchem.5b01198. Epub 2015 Nov 9. J Med Chem. 2016. PMID: 26512410 Review.

2

Small Macrocycles As Highly Active Integrin α2β1 Antagonists.

Halland N, Blum H, Buning C, Kohlmann M, Lindenschmidt A. Halland N, et al. ACS Med Chem Lett. 2014 Jan 10;5(2):193-8. doi: 10.1021/ml4004556. eCollection 2014 Feb 13. ACS Med Chem Lett. 2014. PMID: 24900800 Free PMC article.

3

Rational Design of Highly Potent, Selective, and Bioavailable SGK1 Protein Kinase Inhibitors for the Treatment of Osteoarthritis.

Halland N, Schmidt F, Weiss T, Li Z, Czech J, Saas J, Ding-Pfennigdorff D, Dreyer MK, Strübing C, Nazare M. Halland N, et al. J Med Chem. 2022 Jan 27;65(2):1567-1584. doi: 10.1021/acs.jmedchem.1c01601. Epub 2021 Dec 21. J Med Chem. 2022. PMID: 34931844

4

Discovery of N-[4-(1H-Pyrazolo[3,4-b]pyrazin-6-yl)-phenyl]-sulfonamides as Highly Active and Selective SGK1 Inhibitors.

Halland N, Schmidt F, Weiss T, Saas J, Li Z, Czech J, Dreyer M, Hofmeister A, Mertsch K, Dietz U, Strübing C, Nazare M. Halland N, et al. ACS Med Chem Lett. 2014 Oct 23;6(1):73-8. doi: 10.1021/ml5003376. eCollection 2015 Jan 8. ACS Med Chem Lett. 2014. PMID: 25589934 Free PMC article.

5

Sulfamide as Zinc Binding Motif in Small Molecule Inhibitors of Activated Thrombin Activatable Fibrinolysis Inhibitor (TAFIa).

Halland N, Czech J, Czechtizky W, Evers A, Follmann M, Kohlmann M, Schreuder HA, Kallus C. Halland N, et al. J Med Chem. 2016 Oct 27;59(20):9567-9573. doi: 10.1021/acs.jmedchem.6b01276. Epub 2016 Oct 17. J Med Chem. 2016. PMID: 27749053

6

Novel Small Molecule Inhibitors of Activated Thrombin Activatable Fibrinolysis Inhibitor (TAFIa) from Natural Product Anabaenopeptin.

Halland N, Brönstrup M, Czech J, Czechtizky W, Evers A, Follmann M, Kohlmann M, Schiell M, Kurz M, Schreuder HA, Kallus C. Halland N, et al. J Med Chem. 2015 Jun 11;58(11):4839-44. doi: 10.1021/jm501840b. Epub 2015 May 20. J Med Chem. 2015. PMID: 25990761

7

A general palladium-catalyzed sonogashira coupling of aryl and heteroaryl tosylates.

R'kyek O, Halland N, Lindenschmidt A, Alonso J, Lindemann P, Urmann M, Nazaré M. R'kyek O, et al. Among authors: halland n. Chemistry. 2010 Sep 3;16(33):9986-9. doi: 10.1002/chem.201001524. Chemistry. 2010. PMID: 20607775 No abstract available.

8

The use of virtual screening and differential scanning fluorimetry for the rapid identification of fragments active against MEK1.

Amaning K, Lowinski M, Vallee F, Steier V, Marcireau C, Ugolini A, Delorme C, Foucalt F, McCort G, Derimay N, Andouche C, Vougier S, Llopart S, Halland N, Rak A. Amaning K, et al. Among authors: halland n. Bioorg Med Chem Lett. 2013 Jun 15;23(12):3620-6. doi: 10.1016/j.bmcl.2013.04.003. Epub 2013 Apr 10. Bioorg Med Chem Lett. 2013. PMID: 23648182

9

A general and mild palladium-catalyzed domino reaction for the synthesis of 2H-indazoles.

Halland N, Nazaré M, R'kyek O, Alonso J, Urmann M, Lindenschmidt A. Halland N, et al. Angew Chem Int Ed Engl. 2009;48(37):6879-82. doi: 10.1002/anie.200902323. Angew Chem Int Ed Engl. 2009. PMID: 19681082 No abstract available.

10

A general and mild domino approach to substituted 1-aminoindoles.

Halland N, Nazaré M, Alonso J, R'kyek O, Lindenschmidt A. Halland N, et al. Chem Commun (Camb). 2011 Jan 21;47(3):1042-4. doi: 10.1039/c0cc03584j. Epub 2010 Nov 12. Chem Commun (Camb). 2011. PMID: 21076730

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