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Development and structural analysis of adenosine site binding tankyrase inhibitors.
Bioorg Med Chem Lett. 2016 Jan 15;26(2):328-333. doi: 10.1016/j.bmcl.2015.12.018. Epub 2015 Dec 8.
Bioorg Med Chem Lett. 2016.
PMID: 26706174
Free article.
Structural basis and selectivity of tankyrase inhibition by a Wnt signaling inhibitor WIKI4.
Haikarainen T, Venkannagari H, Narwal M, Obaji E, Lee HW, Nkizinkiko Y, Lehtiö L.
Haikarainen T, et al. Among authors: nkizinkiko y.
PLoS One. 2013 Jun 6;8(6):e65404. doi: 10.1371/journal.pone.0065404. Print 2013.
PLoS One. 2013.
PMID: 23762361
Free PMC article.
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Discovery of potent and selective nonplanar tankyrase inhibiting nicotinamide mimics.
Nkizinkiko Y, Suneel Kumar BVS, Jeankumar VU, Haikarainen T, Koivunen J, Madhuri C, Yogeeswari P, Venkannagari H, Obaji E, Pihlajaniemi T, Sriram D, Lehtiö L.
Nkizinkiko Y, et al.
Bioorg Med Chem. 2015 Aug 1;23(15):4139-4149. doi: 10.1016/j.bmc.2015.06.063. Epub 2015 Jul 2.
Bioorg Med Chem. 2015.
PMID: 26183543
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Discovery of a Novel Series of Tankyrase Inhibitors by a Hybridization Approach.
Anumala UR, Waaler J, Nkizinkiko Y, Ignatev A, Lazarow K, Lindemann P, Olsen PA, Murthy S, Obaji E, Majouga AG, Leonov S, von Kries JP, Lehtiö L, Krauss S, Nazaré M.
Anumala UR, et al. Among authors: nkizinkiko y.
J Med Chem. 2017 Dec 28;60(24):10013-10025. doi: 10.1021/acs.jmedchem.7b00883. Epub 2017 Dec 8.
J Med Chem. 2017.
PMID: 29155568
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2-Phenylquinazolinones as dual-activity tankyrase-kinase inhibitors.
Nkizinkiko Y, Desantis J, Koivunen J, Haikarainen T, Murthy S, Sancineto L, Massari S, Ianni F, Obaji E, Loza MI, Pihlajaniemi T, Brea J, Tabarrini O, Lehtiö L.
Nkizinkiko Y, et al.
Sci Rep. 2018 Jan 26;8(1):1680. doi: 10.1038/s41598-018-19872-3.
Sci Rep. 2018.
PMID: 29374194
Free PMC article.
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Sugar-decorated mesoporous silica nanoparticles as delivery vehicles for the poorly soluble drug celastrol enables targeted induction of apoptosis in cancer cells.
Niemelä E, Desai D, Nkizinkiko Y, Eriksson JE, Rosenholm JM.
Niemelä E, et al. Among authors: nkizinkiko y.
Eur J Pharm Biopharm. 2015 Oct;96:11-21. doi: 10.1016/j.ejpb.2015.07.009. Epub 2015 Jul 14.
Eur J Pharm Biopharm. 2015.
PMID: 26184689
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