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Tetrahydroprotoberberine alkaloids with dopamine and σ receptor affinity.
Bioorg Med Chem. 2016 May 1;24(9):2060-71. doi: 10.1016/j.bmc.2016.03.037. Epub 2016 Mar 21.
Bioorg Med Chem. 2016.
PMID: 27032890
Free PMC article.
Synthesis and evaluation of aporphine analogs containing C1 allyl isosteres at the h5-HT(2A) receptor.
Ponnala S, Kapadia N, Madapa S, Alberts IL, Harding WW.
Ponnala S, et al. Among authors: madapa s.
Bioorg Med Chem Lett. 2015 Nov 15;25(22):5102-6. doi: 10.1016/j.bmcl.2015.10.012. Epub 2015 Oct 9.
Bioorg Med Chem Lett. 2015.
PMID: 26475518
Free PMC article.
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Synthesis and evaluation of C9 alkoxy analogues of (-)-stepholidine as dopamine receptor ligands.
Madapa S, Gadhiya S, Kurtzman T, Alberts IL, Ramsey S, Reith M, Harding WW.
Madapa S, et al.
Eur J Med Chem. 2017 Jan 5;125:255-268. doi: 10.1016/j.ejmech.2016.09.036. Epub 2016 Sep 14.
Eur J Med Chem. 2017.
PMID: 27688181
Free PMC article.
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Semisynthetic Studies on and Biological Evaluation of N-Methyllaurotetanine Analogues as Ligands for 5-HT Receptors.
Madapa S, Harding WW.
Madapa S, et al.
J Nat Prod. 2015 Apr 24;78(4):722-9. doi: 10.1021/np500893h. Epub 2015 Feb 19.
J Nat Prod. 2015.
PMID: 25695425
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Semisynthetic Transformations on (+)-Boldine Reveal a 5-HT2A/2CR Antagonist.
Namballa HK, Madapa S, Sigalapalli DK, Harding WW.
Namballa HK, et al. Among authors: madapa s.
J Nat Prod. 2022 Sep 23;85(9):2149-2158. doi: 10.1021/acs.jnatprod.2c00365. Epub 2022 Aug 24.
J Nat Prod. 2022.
PMID: 36001775
Review.
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Search for new pharmacophores for antimalarial activity. Part II: synthesis and antimalarial activity of new 6-ureido-4-anilinoquinazolines.
Madapa S, Tusi Z, Mishra A, Srivastava K, Pandey SK, Tripathi R, Puri SK, Batra S.
Madapa S, et al.
Bioorg Med Chem. 2009 Jan 1;17(1):222-34. doi: 10.1016/j.bmc.2008.11.005. Epub 2008 Nov 8.
Bioorg Med Chem. 2009.
PMID: 19041250
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Search for new pharmacophores for antimalarial activity. Part I: synthesis and antimalarial activity of new 2-methyl-6-ureido-4-quinolinamides.
Madapa S, Tusi Z, Sridhar D, Kumar A, Siddiqi MI, Srivastava K, Rizvi A, Tripathi R, Puri SK, Shiva Keshava GB, Shukla PK, Batra S.
Madapa S, et al.
Bioorg Med Chem. 2009 Jan 1;17(1):203-21. doi: 10.1016/j.bmc.2008.11.021. Epub 2008 Nov 18.
Bioorg Med Chem. 2009.
PMID: 19058973
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Discovery of MAP855, an Efficacious and Selective MEK1/2 Inhibitor with an ATP-Competitive Mode of Action.
Poddutoori R, Aardalen K, Aithal K, Barahagar SS, Belliappa C, Bock M, Chelur S, Gerken A, Gopinath S, Gruenenfelder B, Kiffe M, Krishnaswami M, Langowski J, Madapa S, Narayanan K, Pandit C, Panigrahi SK, Perrone M, Potakamuri RK, Ramachandra M, Ramanathan A, Ramos R, Sager E, Samajdar S, Subramanya HS, Thimmasandra DS, Venetsanakos E, Möbitz H.
Poddutoori R, et al. Among authors: madapa s.
J Med Chem. 2022 Mar 10;65(5):4350-4366. doi: 10.1021/acs.jmedchem.1c02192. Epub 2022 Feb 23.
J Med Chem. 2022.
PMID: 35195996
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