Kocan M - Search Results

1

ML290 is a biased allosteric agonist at the relaxin receptor RXFP1.

Kocan M, Sarwar M, Ang SY, Xiao J, Marugan JJ, Hossain MA, Wang C, Hutchinson DS, Samuel CS, Agoulnik AI, Bathgate RAD, Summers RJ. Kocan M, et al. Sci Rep. 2017 Jun 7;7(1):2968. doi: 10.1038/s41598-017-02916-5. Sci Rep. 2017. PMID: 28592882 Free PMC article.

2

β(2)-Adrenoceptors increase translocation of GLUT4 via GPCR kinase sites in the receptor C-terminal tail.

Dehvari N, Hutchinson DS, Nevzorova J, Dallner OS, Sato M, Kocan M, Merlin J, Evans BA, Summers RJ, Bengtsson T. Dehvari N, et al. Among authors: kocan m. Br J Pharmacol. 2012 Mar;165(5):1442-56. doi: 10.1111/j.1476-5381.2011.01647.x. Br J Pharmacol. 2012. PMID: 21883150 Free PMC article.

3

Minimization of human relaxin-3 leading to high-affinity analogues with increased selectivity for relaxin-family peptide 3 receptor (RXFP3) over RXFP1.

Shabanpoor F, Akhter Hossain M, Ryan PJ, Belgi A, Layfield S, Kocan M, Zhang S, Samuel CS, Gundlach AL, Bathgate RA, Separovic F, Wade JD. Shabanpoor F, et al. Among authors: kocan m. J Med Chem. 2012 Feb 23;55(4):1671-81. doi: 10.1021/jm201505p. Epub 2012 Feb 8. J Med Chem. 2012. PMID: 22257012

4

Relaxin family peptides and their receptors.

Bathgate RA, Halls ML, van der Westhuizen ET, Callander GE, Kocan M, Summers RJ. Bathgate RA, et al. Among authors: kocan m. Physiol Rev. 2013 Jan;93(1):405-80. doi: 10.1152/physrev.00001.2012. Physiol Rev. 2013. PMID: 23303914 Free article. Review.

5

Minimum active structure of insulin-like peptide 5.

Belgi A, Bathgate RA, Kocan M, Patil N, Zhang S, Tregear GW, Wade JD, Hossain MA. Belgi A, et al. Among authors: kocan m. J Med Chem. 2013 Dec 12;56(23):9509-16. doi: 10.1021/jm400924p. Epub 2013 Nov 21. J Med Chem. 2013. PMID: 24188028

6

Relaxin requires the angiotensin II type 2 receptor to abrogate renal interstitial fibrosis.

Chow BS, Kocan M, Bosnyak S, Sarwar M, Wigg B, Jones ES, Widdop RE, Summers RJ, Bathgate RA, Hewitson TD, Samuel CS. Chow BS, et al. Among authors: kocan m. Kidney Int. 2014 Jul;86(1):75-85. doi: 10.1038/ki.2013.518. Epub 2014 Jan 15. Kidney Int. 2014. PMID: 24429402 Free article.

7

Signalling profiles of H3 relaxin, H2 relaxin and R3(BΔ23-27)R/I5 acting at the relaxin family peptide receptor 3 (RXFP3).

Kocan M, Sarwar M, Hossain MA, Wade JD, Summers RJ. Kocan M, et al. Br J Pharmacol. 2014 Jun;171(11):2827-41. doi: 10.1111/bph.12623. Br J Pharmacol. 2014. PMID: 24641548 Free PMC article.

8

Orthosteric, Allosteric and Biased Signalling at the Relaxin-3 Receptor RXFP3.

Kocan M, Ang SY, Summers RJ. Kocan M, et al. Neurochem Res. 2016 Mar;41(3):610-9. doi: 10.1007/s11064-015-1701-3. Epub 2015 Aug 21. Neurochem Res. 2016. PMID: 26294284

9

The C-terminus of the B-chain of human insulin-like peptide 5 is critical for cognate RXFP4 receptor activity.

Patil NA, Bathgate RAD, Kocan M, Ang SY, Tailhades J, Separovic F, Summers R, Grosse J, Hughes RA, Wade JD, Hossain MA. Patil NA, et al. Among authors: kocan m. Amino Acids. 2016 Apr;48(4):987-992. doi: 10.1007/s00726-015-2144-5. Epub 2015 Dec 11. Amino Acids. 2016. PMID: 26661035

10

Engineering of a Novel Simplified Human Insulin-Like Peptide 5 Agonist.

Patil NA, Hughes RA, Rosengren KJ, Kocan M, Ang SY, Tailhades J, Separovic F, Summers RJ, Grosse J, Wade JD, Bathgate RA, Hossain MA. Patil NA, et al. Among authors: kocan m. J Med Chem. 2016 Mar 10;59(5):2118-25. doi: 10.1021/acs.jmedchem.5b01786. Epub 2016 Feb 12. J Med Chem. 2016. PMID: 26824523

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