Search Page
Save citations to file
Email citations
Send citations to clipboard
Add to Collections
Add to My Bibliography
Create a file for external citation management software
Your saved search
Your RSS Feed
Search Results
7 results
Filters applied: . Clear all
Results are displayed in a computed author sort order.
The Results By Year timeline is not available.
Page 1
Discovery of Highly Potent and Selective Small-Molecule Reversible Factor D Inhibitors Demonstrating Alternative Complement Pathway Inhibition in Vivo.
J Med Chem. 2017 Jul 13;60(13):5717-5735. doi: 10.1021/acs.jmedchem.7b00425. Epub 2017 Jun 30.
J Med Chem. 2017.
PMID: 28621538
Small-molecule factor D inhibitors targeting the alternative complement pathway.
Maibaum J, Liao SM, Vulpetti A, Ostermann N, Randl S, Rüdisser S, Lorthiois E, Erbel P, Kinzel B, Kolb FA, Barbieri S, Wagner J, Durand C, Fettis K, Dussauge S, Hughes N, Delgado O, Hommel U, Gould T, Mac Sweeney A, Gerhartz B, Cumin F, Flohr S, Schubart A, Jaffee B, Harrison R, Risitano AM, Eder J, Anderson K.
Maibaum J, et al. Among authors: fettis k.
Nat Chem Biol. 2016 Dec;12(12):1105-1110. doi: 10.1038/nchembio.2208. Epub 2016 Oct 24.
Nat Chem Biol. 2016.
PMID: 27775713
Item in Clipboard
Structure-Based Design and Preclinical Characterization of Selective and Orally Bioavailable Factor XIa Inhibitors: Demonstrating the Power of an Integrated S1 Protease Family Approach.
Lorthiois E, Roache J, Barnes-Seeman D, Altmann E, Hassiepen U, Turner G, Duvadie R, Hornak V, Karki RG, Schiering N, Weihofen WA, Perruccio F, Calhoun A, Fazal T, Dedic D, Durand C, Dussauge S, Fettis K, Tritsch F, Dentel C, Druet A, Liu D, Kirman L, Lachal J, Namoto K, Bevan D, Mo R, Monnet G, Muller L, Zessis R, Huang X, Lindsley L, Currie T, Chiu YH, Fridrich C, Delgado P, Wang S, Hollis-Symynkywicz M, Berghausen J, Williams E, Liu H, Liang G, Kim H, Hoffmann P, Hein A, Ramage P, D'Arcy A, Harlfinger S, Renatus M, Ruedisser S, Feldman D, Elliott J, Sedrani R, Maibaum J, Adams CM.
Lorthiois E, et al. Among authors: fettis k.
J Med Chem. 2020 Aug 13;63(15):8088-8113. doi: 10.1021/acs.jmedchem.0c00279. Epub 2020 Jul 21.
J Med Chem. 2020.
PMID: 32551603
Item in Clipboard
Trithiocarbonates as a novel class of HDAC inhibitors: SAR studies, isoenzyme selectivity, and pharmacological profiles.
Dehmel F, Weinbrenner S, Julius H, Ciossek T, Maier T, Stengel T, Fettis K, Burkhardt C, Wieland H, Beckers T.
Dehmel F, et al. Among authors: fettis k.
J Med Chem. 2008 Jul 10;51(13):3985-4001. doi: 10.1021/jm800093c. Epub 2008 Jun 18.
J Med Chem. 2008.
PMID: 18558669
Item in Clipboard
Self-assembly of noncyclic bis-D- and L-tripeptides into higher order tubular constructs: design, synthesis, and X-ray crystal superstructure.
Hanessian S, Vinci V, Fettis K, Maris T, Viet MT.
Hanessian S, et al. Among authors: fettis k.
J Org Chem. 2008 Feb 15;73(4):1181-91. doi: 10.1021/jo701621c. Epub 2007 Dec 7.
J Org Chem. 2008.
PMID: 18062697
Item in Clipboard
Synthesis of 3 10-helix-inducing constrained analogues of L-proline.
Hanessian S, Papeo G, Fettis K, Therrien E, Viet MT.
Hanessian S, et al. Among authors: fettis k.
J Org Chem. 2004 Jul 23;69(15):4891-9. doi: 10.1021/jo0401422.
J Org Chem. 2004.
PMID: 15255713
Item in Clipboard
Synthesis of functionally diverse and conformationally constrained polycyclic analogues of proline and prolinol.
Hanessian S, Papeo G, Angiolini M, Fettis K, Beretta M, Munro A.
Hanessian S, et al. Among authors: fettis k.
J Org Chem. 2003 Sep 19;68(19):7204-18. doi: 10.1021/jo0301447.
J Org Chem. 2003.
PMID: 12968869
Item in Clipboard
Cite
Cite