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Discovery of potent and selective inhibitors of calmodulin-dependent kinase II (CaMKII).
Bioorg Med Chem Lett. 2018 Feb 1;28(3):541-546. doi: 10.1016/j.bmcl.2017.10.040. Epub 2017 Oct 20.
Bioorg Med Chem Lett. 2018.
PMID: 29254643
Prodrugs of a 1'-CN-4-Aza-7,9-dideazaadenosine C-Nucleoside Leading to the Discovery of Remdesivir (GS-5734) as a Potent Inhibitor of Respiratory Syncytial Virus with Efficacy in the African Green Monkey Model of RSV.
Mackman RL, Hui HC, Perron M, Murakami E, Palmiotti C, Lee G, Stray K, Zhang L, Goyal B, Chun K, Byun D, Siegel D, Simonovich S, Du Pont V, Pitts J, Babusis D, Vijjapurapu A, Lu X, Kim C, Zhao X, Chan J, Ma B, Lye D, Vandersteen A, Wortman S, Barrett KT, Toteva M, Jordan R, Subramanian R, Bilello JP, Cihlar T.
Mackman RL, et al.
J Med Chem. 2021 Apr 22;64(8):5001-5017. doi: 10.1021/acs.jmedchem.1c00071. Epub 2021 Apr 9.
J Med Chem. 2021.
PMID: 33835812
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Discovery and in Vivo Evaluation of Macrocyclic Mcl-1 Inhibitors Featuring an α-Hydroxy Phenylacetic Acid Pharmacophore or Bioisostere.
Rescourio G, Gonzalez AZ, Jabri S, Belmontes B, Moody G, Whittington D, Huang X, Caenepeel S, Cardozo M, Cheng AC, Chow D, Dou H, Jones A, Kelly RC, Li Y, Lizarzaburu M, Lo MC, Mallari R, Meleza C, Rew Y, Simonovich S, Sun D, Turcotte S, Yan X, Wong SG, Yanez E, Zancanella M, Houze J, Medina JC, Hughes PE, Brown SP.
Rescourio G, et al. Among authors: simonovich s.
J Med Chem. 2019 Nov 27;62(22):10258-10271. doi: 10.1021/acs.jmedchem.9b01310. Epub 2019 Nov 18.
J Med Chem. 2019.
PMID: 31736296
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A general approach to the enantioselective α-oxidation of aldehydes via synergistic catalysis.
Simonovich SP, Van Humbeck JF, Macmillan DW.
Simonovich SP, et al.
Chem Sci. 2012;3(1):58-61. doi: 10.1039/c1sc00556a.
Chem Sci. 2012.
PMID: 22308217
Free PMC article.
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Enantioselective α-arylation of carbonyls via Cu(I)-bisoxazoline catalysis.
Harvey JS, Simonovich SP, Jamison CR, MacMillan DW.
Harvey JS, et al. Among authors: simonovich sp.
J Am Chem Soc. 2011 Sep 7;133(35):13782-5. doi: 10.1021/ja206050b. Epub 2011 Aug 17.
J Am Chem Soc. 2011.
PMID: 21848265
Free PMC article.
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Concerning the mechanism of the FeCl3-catalyzed alpha-oxyamination of aldehydes: evidence for a non-SOMO activation pathway.
Van Humbeck JF, Simonovich SP, Knowles RR, MacMillan DW.
Van Humbeck JF, et al. Among authors: simonovich sp.
J Am Chem Soc. 2010 Jul 28;132(29):10012-4. doi: 10.1021/ja1043006.
J Am Chem Soc. 2010.
PMID: 20608675
Free PMC article.
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