Ghinet A - Search Results

1

Pyroglutamide-Based P2X7 Receptor Antagonists Targeting Inflammatory Bowel Disease.

Homerin G, Jawhara S, Dezitter X, Baudelet D, Dufrénoy P, Rigo B, Millet R, Furman C, Ragé G, Lipka E, Farce A, Renault N, Sendid B, Charlet R, Leroy J, Phanithavong M, Richeval C, Wiart JF, Allorge D, Adriouch S, Vouret-Craviari V, Ghinet A. Homerin G, et al. Among authors: ghinet a. J Med Chem. 2020 Mar 12;63(5):2074-2094. doi: 10.1021/acs.jmedchem.9b00584. Epub 2019 Sep 27. J Med Chem. 2020. PMID: 31525963

2

In vitro metabolism of phenstatin: potential pharmacological consequences.

Le Broc-Ryckewaert D, Pommery N, Pommery J, Ghinet A, Farce A, Wiart JF, Gautret P, Rigo B, Hénichart JP. Le Broc-Ryckewaert D, et al. Among authors: ghinet a. Drug Metab Lett. 2011 Aug;5(3):209-15. doi: 10.2174/187231211796904973. Drug Metab Lett. 2011. PMID: 21679150

3

Synthesis and biological evaluation of phenstatin metabolites.

Ghinet A, Rigo B, Hénichart JP, Le Broc-Ryckewaert D, Pommery J, Pommery N, Thuru X, Quesnel B, Gautret P. Ghinet A, et al. Bioorg Med Chem. 2011 Oct 15;19(20):6042-54. doi: 10.1016/j.bmc.2011.08.047. Epub 2011 Aug 27. Bioorg Med Chem. 2011. PMID: 21920767

4

New farnesyltransferase inhibitors in the phenothiazine series.

Belei D, Dumea C, Samson A, Farce A, Dubois J, Bîcu E, Ghinet A. Belei D, et al. Among authors: ghinet a. Bioorg Med Chem Lett. 2012 Jul 15;22(14):4517-22. doi: 10.1016/j.bmcl.2012.06.007. Epub 2012 Jun 9. Bioorg Med Chem Lett. 2012. PMID: 22738631

5

Antioxidant activity of new benzo[de]quinolines and lactams: 2D-quantitative structure-activity relationships.

Ghinet A, Farce A, Oudir S, Pommery J, Vamecq J, Henichart JP, Rigo B, Gautret P. Ghinet A, et al. Med Chem. 2012 Sep;8(5):942-6. doi: 10.2174/157340612802084216. Med Chem. 2012. PMID: 22741798

6

Synthesis and biological evaluation of new phenothiazine derivatives bearing a pyrazole unit as protein farnesyltransferase inhibitors.

Baciu-Atudosie L, Ghinet A, Farce A, Dubois J, Belei D, Bîcu E. Baciu-Atudosie L, et al. Among authors: ghinet a. Bioorg Med Chem Lett. 2012 Nov 15;22(22):6896-902. doi: 10.1016/j.bmcl.2012.09.030. Epub 2012 Sep 17. Bioorg Med Chem Lett. 2012. PMID: 23036952

7

Synthesis and anticancer activity of analogues of phenstatin, with a phenothiazine A-ring, as a new class of microtubule-targeting agents.

Abuhaie CM, Bîcu E, Rigo B, Gautret P, Belei D, Farce A, Dubois J, Ghinet A. Abuhaie CM, et al. Among authors: ghinet a. Bioorg Med Chem Lett. 2013 Jan 1;23(1):147-52. doi: 10.1016/j.bmcl.2012.10.135. Epub 2012 Nov 8. Bioorg Med Chem Lett. 2013. PMID: 23200248

8

Synthesis and biological evaluation of a new series of phenothiazine-containing protein farnesyltransferase inhibitors.

Abuhaie CM, Ghinet A, Farce A, Dubois J, Gautret P, Rigo B, Belei D, Bîcu E. Abuhaie CM, et al. Among authors: ghinet a. Eur J Med Chem. 2013 Jan;59:101-10. doi: 10.1016/j.ejmech.2012.11.008. Epub 2012 Nov 14. Eur J Med Chem. 2013. PMID: 23207411

9

Synthesis and biological evaluation of fluoro analogues of antimitotic phenstatin.

Ghinet A, Tourteau A, Rigo B, Stocker V, Leman M, Farce A, Dubois J, Gautret P. Ghinet A, et al. Bioorg Med Chem. 2013 Jun 1;21(11):2932-40. doi: 10.1016/j.bmc.2013.03.064. Epub 2013 Apr 4. Bioorg Med Chem. 2013. PMID: 23618708

10

Synthesis and biological evaluation of a new series of N-ylides as protein farnesyltransferase inhibitors.

Abuhaie CM, Ghinet A, Farce A, Dubois J, Rigo B, Bîcu E. Abuhaie CM, et al. Among authors: ghinet a. Bioorg Med Chem Lett. 2013 Nov 1;23(21):5887-92. doi: 10.1016/j.bmcl.2013.08.088. Epub 2013 Sep 3. Bioorg Med Chem Lett. 2013. PMID: 24054122

Save citations to file

Email citations

Send citations to clipboard

Add to Collections

Add to My Bibliography

Create a file for external citation management software

Your saved search

Your RSS Feed

My NCBI Filters

Text availability

Article attribute

Article type

Publication date

66 results

Search Page