Millet R - Search Results

1

Pyroglutamide-Based P2X7 Receptor Antagonists Targeting Inflammatory Bowel Disease.

Homerin G, Jawhara S, Dezitter X, Baudelet D, Dufrénoy P, Rigo B, Millet R, Furman C, Ragé G, Lipka E, Farce A, Renault N, Sendid B, Charlet R, Leroy J, Phanithavong M, Richeval C, Wiart JF, Allorge D, Adriouch S, Vouret-Craviari V, Ghinet A. Homerin G, et al. Among authors: millet r. J Med Chem. 2020 Mar 12;63(5):2074-2094. doi: 10.1021/acs.jmedchem.9b00584. Epub 2019 Sep 27. J Med Chem. 2020. PMID: 31525963

2

Novel potent substance P and neurokinin A receptor antagonists. Conception, synthesis and biological evaluation of indolizine derivatives.

Millet R, Domarkas J, Rigo B, Goossens L, Goossens JF, Houssin R, Hénichart JP. Millet R, et al. Bioorg Med Chem. 2002 Sep;10(9):2905-12. doi: 10.1016/s0968-0896(02)00144-x. Bioorg Med Chem. 2002. PMID: 12110311

3

Potent and selective farnesyl transferase inhibitors.

Millet R, Domarkas J, Houssin R, Gilleron P, Goossens JF, Chavatte P, Logé C, Pommery N, Pommery J, Hénichart JP. Millet R, et al. J Med Chem. 2004 Dec 30;47(27):6812-20. doi: 10.1021/jm030502y. J Med Chem. 2004. PMID: 15615530

4

Synthesis of a novel conformationally restricted Val-Phe dipeptidomimetic.

Gilleron P, Millet R, Domarkas J, Farce A, Houssin R, Hénichart JP. Gilleron P, et al. Among authors: millet r. J Pept Sci. 2006 Feb;12(2):140-6. doi: 10.1002/psc.688. J Pept Sci. 2006. PMID: 15948143

5

Novel 4-oxo-1,4-dihydroquinoline-3-carboxamide derivatives as new CB2 cannabinoid receptors agonists: synthesis, pharmacological properties and molecular modeling.

Stern E, Muccioli GG, Millet R, Goossens JF, Farce A, Chavatte P, Poupaert JH, Lambert DM, Depreux P, Hénichart JP. Stern E, et al. Among authors: millet r. J Med Chem. 2006 Jan 12;49(1):70-9. doi: 10.1021/jm050467q. J Med Chem. 2006. PMID: 16392793

6

Solid-phase synthesis and pharmacological evaluation of a library of peptidomimetics as potential farnesyltransferase inhibitors: an approach to new lead compounds.

Gilleron P, Millet R, Houssin R, Wlodarczyk N, Farce A, Lemoine A, Goossens JF, Chavatte P, Pommery N, Hénichart JP. Gilleron P, et al. Among authors: millet r. Eur J Med Chem. 2006 Jun;41(6):745-55. doi: 10.1016/j.ejmech.2006.03.017. Epub 2006 May 2. Eur J Med Chem. 2006. PMID: 16647166

7

Design, synthesis and biological evaluation of substituted dioxodibenzothiazepines and dibenzocycloheptanes as farnesyltransferase inhibitors.

Gilleron P, Wlodarczyk N, Houssin R, Farce A, Laconde G, Goossens JF, Lemoine A, Pommery N, Hénichart JP, Millet R. Gilleron P, et al. Among authors: millet r. Bioorg Med Chem Lett. 2007 Oct 1;17(19):5465-71. doi: 10.1016/j.bmcl.2007.07.002. Epub 2007 Jul 7. Bioorg Med Chem Lett. 2007. PMID: 17827015

8

Pharmacomodulations around the 4-oxo-1,4-dihydroquinoline-3-carboxamides, a class of potent CB2-selective cannabinoid receptor ligands: consequences in receptor affinity and functionality.

Stern E, Muccioli GG, Bosier B, Hamtiaux L, Millet R, Poupaert JH, Hénichart JP, Depreux P, Goossens JF, Lambert DM. Stern E, et al. Among authors: millet r. J Med Chem. 2007 Nov 1;50(22):5471-84. doi: 10.1021/jm070387h. Epub 2007 Oct 4. J Med Chem. 2007. PMID: 17915849

9

4-Oxo-1,4-dihydropyridines as selective CB2 cannabinoid receptor ligands: structural insights into the design of a novel inverse agonist series.

El Bakali J, Muccioli GG, Renault N, Pradal D, Body-Malapel M, Djouina M, Hamtiaux L, Andrzejak V, Desreumaux P, Chavatte P, Lambert DM, Millet R. El Bakali J, et al. Among authors: millet r. J Med Chem. 2010 Nov 25;53(22):7918-31. doi: 10.1021/jm100286k. Epub 2010 Oct 27. J Med Chem. 2010. PMID: 20979417

10

Potent farnesyltransferase inhibitors with 1,4-diazepane scaffolds as novel destabilizing microtubule agents in hormone-resistant prostate cancer.

Wlodarczyk N, Le Broc-Ryckewaert D, Gilleron P, Lemoine A, Farce A, Chavatte P, Dubois J, Pommery N, Hénichart JP, Furman C, Millet R. Wlodarczyk N, et al. Among authors: millet r. J Med Chem. 2011 Mar 10;54(5):1178-90. doi: 10.1021/jm101067y. Epub 2011 Feb 7. J Med Chem. 2011. PMID: 21299244

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