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Design, Synthesis, and Pharmacological Characterization of a Neutral, Non-Prodrug Thrombin Inhibitor with Good Oral Pharmacokinetics.
J Med Chem. 2020 Nov 12;63(21):12574-12594. doi: 10.1021/acs.jmedchem.0c01035. Epub 2020 Oct 27.
J Med Chem. 2020.
PMID: 33108181
Free article.
Discovery and Characterization of the Potent and Selective P2X4 Inhibitor N-[4-(3-Chlorophenoxy)-3-sulfamoylphenyl]-2-phenylacetamide (BAY-1797) and Structure-Guided Amelioration of Its CYP3A4 Induction Profile.
Werner S, Mesch S, Hillig RC, Ter Laak A, Klint J, Neagoe I, Laux-Biehlmann A, Dahllöf H, Bräuer N, Puetter V, Nubbemeyer R, Schulz S, Bairlein M, Zollner TM, Steinmeyer A.
Werner S, et al. Among authors: puetter v.
J Med Chem. 2019 Dec 26;62(24):11194-11217. doi: 10.1021/acs.jmedchem.9b01304. Epub 2019 Dec 11.
J Med Chem. 2019.
PMID: 31746599
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Novel small molecule inhibitors of MDR Mycobacterium tuberculosis by NMR fragment screening of antigen 85C.
Scheich C, Puetter V, Schade M.
Scheich C, et al. Among authors: puetter v.
J Med Chem. 2010 Dec 9;53(23):8362-7. doi: 10.1021/jm100993z. Epub 2010 Nov 12.
J Med Chem. 2010.
PMID: 21073150
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Functional and Structural Characterization of Bub3·BubR1 Interactions Required for Spindle Assembly Checkpoint Signaling in Human Cells.
Prinz F, Puetter V, Holton SJ, Andres D, Stegmann CM, Kwiatkowski D, Prechtl S, Petersen K, Beckmann G, Kreft B, Mumberg D, Fernández-Montalván A.
Prinz F, et al. Among authors: puetter v.
J Biol Chem. 2016 May 20;291(21):11252-67. doi: 10.1074/jbc.M115.702142. Epub 2016 Mar 30.
J Biol Chem. 2016.
PMID: 27030009
Free PMC article.
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Isoform-Selective ATAD2 Chemical Probe with Novel Chemical Structure and Unusual Mode of Action.
Fernández-Montalván AE, Berger M, Kuropka B, Koo SJ, Badock V, Weiske J, Puetter V, Holton SJ, Stöckigt D, Ter Laak A, Centrella PA, Clark MA, Dumelin CE, Sigel EA, Soutter HH, Troast DM, Zhang Y, Cuozzo JW, Keefe AD, Roche D, Rodeschini V, Chaikuad A, Díaz-Sáez L, Bennett JM, Fedorov O, Huber KVM, Hübner J, Weinmann H, Hartung IV, Gorjánácz M.
Fernández-Montalván AE, et al. Among authors: puetter v.
ACS Chem Biol. 2017 Nov 17;12(11):2730-2736. doi: 10.1021/acschembio.7b00708. Epub 2017 Oct 24.
ACS Chem Biol. 2017.
PMID: 29043777
Free PMC article.
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A dual estrogen receptor TR-FRET assay for simultaneous measurement of steroid site binding and coactivator recruitment.
Hilal T, Puetter V, Otto C, Parczyk K, Bader B.
Hilal T, et al. Among authors: puetter v.
J Biomol Screen. 2010 Mar;15(3):268-78. doi: 10.1177/1087057109359196. Epub 2010 Feb 11.
J Biomol Screen. 2010.
PMID: 20150592
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High-Throughput Expression and Purification of Human Solute Carriers for Structural and Biochemical Studies.
Raturi S, Li H, Chang YN, Scacioc A, Bohstedt T, Fernandez-Cid A, Evans A, Abrusci P, Balakrishnan A, Pascoa TC, He D, Chi G, Kaur Singh N, Ye M, Li A, Shrestha L, Wang D, Williams EP, Burgess-Brown NA, Dürr KL, Puetter V, Ingles-Prieto A, Sauer DB.
Raturi S, et al. Among authors: puetter v.
J Vis Exp. 2023 Sep 29;(199). doi: 10.3791/65878.
J Vis Exp. 2023.
PMID: 37843272
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