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Development of a 1,2,4-Triazole-Based Lead Tankyrase Inhibitor: Part II.
J Med Chem. 2021 Dec 23;64(24):17936-17949. doi: 10.1021/acs.jmedchem.1c01264. Epub 2021 Dec 8.
J Med Chem. 2021.
PMID: 34878777
Free PMC article.
Preclinical Lead Optimization of a 1,2,4-Triazole Based Tankyrase Inhibitor.
Waaler J, Leenders RGG, Sowa ST, Alam Brinch S, Lycke M, Nieczypor P, Aertssen S, Murthy S, Galera-Prat A, Damen E, Wegert A, Nazaré M, Lehtiö L, Krauss S.
Waaler J, et al. Among authors: aertssen s.
J Med Chem. 2020 Jul 9;63(13):6834-6846. doi: 10.1021/acs.jmedchem.0c00208. Epub 2020 Jun 23.
J Med Chem. 2020.
PMID: 32511917
Free PMC article.
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Cyclopentitol as a scaffold for a natural product-like compound library for drug discovery.
Padwal JD, Filippov DV, Narhe BD, Aertssen S, Beuving RJ, Benningshof JC, van der Marel GA, Overkleeft HS, van der Stelt M.
Padwal JD, et al. Among authors: aertssen s.
Bioorg Med Chem. 2015 Jun 1;23(11):2650-5. doi: 10.1016/j.bmc.2015.01.040. Epub 2015 Jan 31.
Bioorg Med Chem. 2015.
PMID: 25691210
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