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Mycobactin Analogues with Excellent Pharmacokinetic Profile Demonstrate Potent Antitubercular Specific Activity and Exceptional Efflux Pump Inhibition.
J Med Chem. 2022 Jan 13;65(1):234-256. doi: 10.1021/acs.jmedchem.1c01349. Epub 2022 Jan 4.
J Med Chem. 2022.
PMID: 34981940
Cytotoxic activity of quinolinequinones in cancer: In vitro studies, molecular docking, and ADME/PK profiling.
Jannuzzi AT, Yilmaz Goler AM, Shilkar D, Mondal S, Basavanakatti VN, Yıldırım H, Yıldız M, Çelik Onar H, Bayrak N, Jayaprakash V, TuYuN AF.
Jannuzzi AT, et al. Among authors: basavanakatti vn.
Chem Biol Drug Des. 2023 Nov;102(5):1133-1154. doi: 10.1111/cbdd.14314. Epub 2023 Aug 3.
Chem Biol Drug Des. 2023.
PMID: 37537000
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Analysis of Quinolinequinone Analogs with Promising Cytotoxic Activity against Breast Cancer.
Yilmaz Goler AM, Tarbin Jannuzzi A, Biswas A, Mondal S, Basavanakatti VN, Jayaprakash Venkatesan R, Yıldırım H, Yıldız M, Çelik Onar H, Bayrak N, Jayaprakash V, TuYuN AF.
Yilmaz Goler AM, et al. Among authors: basavanakatti vn.
Chem Biodivers. 2023 Sep;20(9):e202300848. doi: 10.1002/cbdv.202300848. Epub 2023 Aug 23.
Chem Biodivers. 2023.
PMID: 37590495
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Validation of 96-well equilibrium dialysis with non-radiolabeled drug for definitive measurement of protein binding and application to clinical development of highly-bound drugs.
Zamek-Gliszczynski MJ, Ruterbories KJ, Ajamie RT, Wickremsinhe ER, Pothuri L, Rao MV, Basavanakatti VN, Pinjari J, Ramanathan VK, Chaudhary AK.
Zamek-Gliszczynski MJ, et al. Among authors: basavanakatti vn.
J Pharm Sci. 2011 Jun;100(6):2498-507. doi: 10.1002/jps.22452. Epub 2011 Jan 6.
J Pharm Sci. 2011.
PMID: 21213309
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