Intagliata S - Search Results

1

Characterization of CM-398, a Novel Selective Sigma-2 Receptor Ligand, as a Potential Therapeutic for Neuropathic Pain.

Wilson LL, Alleyne AR, Eans SO, Cirino TJ, Stacy HM, Mottinelli M, Intagliata S, McCurdy CR, McLaughlin JP. Wilson LL, et al. Among authors: intagliata s. Molecules. 2022 Jun 4;27(11):3617. doi: 10.3390/molecules27113617. Molecules. 2022. PMID: 35684553 Free PMC article.

2

Novel Structural Insight into Inhibitors of Heme Oxygenase-1 (HO-1) by New Imidazole-Based Compounds: Biochemical and In Vitro Anticancer Activity Evaluation.

Greish KF, Salerno L, Al Zahrani R, Amata E, Modica MN, Romeo G, Marrazzo A, Prezzavento O, Sorrenti V, Rescifina A, Floresta G, Intagliata S, Pittalà V. Greish KF, et al. Among authors: intagliata s. Molecules. 2018 May 18;23(5):1209. doi: 10.3390/molecules23051209. Molecules. 2018. PMID: 29783634 Free PMC article.

3

Divergent Cytotoxic and Metabolically Stimulative Functions of Sigma-2 Receptors: Structure-Activity Relationships of 6-Acetyl-3-(4-(4-(4-fluorophenyl)piperazin-1-yl)butyl)benzo[d]oxazol-2(3H)-one (SN79) Derivatives.

Nicholson HE, Alsharif WF, Comeau AB, Mesangeau C, Intagliata S, Mottinelli M, McCurdy CR, Bowen WD. Nicholson HE, et al. Among authors: intagliata s. J Pharmacol Exp Ther. 2019 Feb;368(2):272-281. doi: 10.1124/jpet.118.253484. Epub 2018 Dec 7. J Pharmacol Exp Ther. 2019. PMID: 30530624 Free PMC article.

4

Benzimidazolone-based selective σ₂ receptor ligands: Synthesis and pharmacological evaluation.

Intagliata S, Alsharif WF, Mesangeau C, Fazio N, Seminerio M, Xu YT, Matsumoto RR, McCurdy CR. Intagliata S, et al. Eur J Med Chem. 2019 Mar 1;165:250-257. doi: 10.1016/j.ejmech.2019.01.019. Epub 2019 Jan 9. Eur J Med Chem. 2019. PMID: 30685525 Free PMC article.

5

Synthesis, in vitro and in vivo characterization of new benzoxazole and benzothiazole-based sigma receptor ligands.

Romeo G, Prezzavento O, Intagliata S, Pittalà V, Modica MN, Marrazzo A, Turnaturi R, Parenti C, Chiechio S, Arena E, Campisi A, Sposito G, Salerno L. Romeo G, et al. Among authors: intagliata s. Eur J Med Chem. 2019 Jul 15;174:226-235. doi: 10.1016/j.ejmech.2019.04.056. Epub 2019 Apr 21. Eur J Med Chem. 2019. PMID: 31042618

6

Characterization of Sigma 1 Receptor Antagonist CM-304 and Its Analog, AZ-66: Novel Therapeutics Against Allodynia and Induced Pain.

Cirino TJ, Eans SO, Medina JM, Wilson LL, Mottinelli M, Intagliata S, McCurdy CR, McLaughlin JP. Cirino TJ, et al. Among authors: intagliata s. Front Pharmacol. 2019 Jun 14;10:678. doi: 10.3389/fphar.2019.00678. eCollection 2019. Front Pharmacol. 2019. PMID: 31258480 Free PMC article.

7

Synthesis and Molecular Modelling Studies of New 1,3-Diaryl-5-Oxo-Proline Derivatives as Endothelin Receptor Ligands.

Intagliata S, Helal MA, Materia L, Pittalà V, Salerno L, Marrazzo A, Cagnotto A, Salmona M, Modica MN, Romeo G. Intagliata S, et al. Molecules. 2020 Apr 17;25(8):1851. doi: 10.3390/molecules25081851. Molecules. 2020. PMID: 32316541 Free PMC article.

8

Discovery of a Highly Selective Sigma-2 Receptor Ligand, 1-(4-(6,7-Dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)butyl)-3-methyl-1H-benzo[d]imidazol-2(3H)-one (CM398), with Drug-Like Properties and Antinociceptive Effects In Vivo.

Intagliata S, Sharma A, King TI, Mesangeau C, Seminerio M, Chin FT, Wilson LL, Matsumoto RR, McLaughlin JP, Avery BA, McCurdy CR. Intagliata S, et al. AAPS J. 2020 Jul 20;22(5):94. doi: 10.1208/s12248-020-00472-x. AAPS J. 2020. PMID: 32691179

9

Bioanalytical method development and pharmacokinetics of MCI-92, a sigma-1 receptor ligand.

Popa R, Kamble SH, Kanumuri RS, King TI, Berthold EC, Intagliata S, Sharma A, McCurdy CR. Popa R, et al. Among authors: intagliata s. J Pharm Biomed Anal. 2020 Nov 30;191:113610. doi: 10.1016/j.jpba.2020.113610. Epub 2020 Sep 13. J Pharm Biomed Anal. 2020. PMID: 32971495

10

Exploring 1-adamantanamine as an alternative amine moiety for metabolically labile azepane ring in newly synthesized benzo[d]thiazol-2(3H)one σ receptor ligands.

Intagliata S, Agha H, Kopajtic TA, Katz JL, Kamble SH, Sharma A, Avery BA, McCurdy CR. Intagliata S, et al. Med Chem Res. 2020 Sep;29(9):1697-1706. doi: 10.1007/s00044-020-02597-2. Epub 2020 Jul 8. Med Chem Res. 2020. PMID: 33584084 Free PMC article.

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