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Pivotal role of nitrogen heterocycles in Alzheimer's disease drug discovery.
Drug Discov Today. 2022 Oct;27(10):103322. doi: 10.1016/j.drudis.2022.07.007. Epub 2022 Jul 19.
Drug Discov Today. 2022.
PMID: 35868626
Review.
Functionalized Allopurinols Targeting Amyloid-Binding Alcohol Dehydrogenase Rescue Aβ-Induced Mitochondrial Dysfunction.
Morsy A, Maddeboina K, Gao J, Wang H, Valdez J, Dow LF, Wang X, Trippier PC.
Morsy A, et al. Among authors: maddeboina k.
ACS Chem Neurosci. 2022 Jul 20;13(14):2176-2190. doi: 10.1021/acschemneuro.2c00246. Epub 2022 Jul 8.
ACS Chem Neurosci. 2022.
PMID: 35802826
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Aldo-Keto Reductase 1C3 Inhibitor Prodrug Improves Pharmacokinetic Profile and Demonstrates In Vivo Efficacy in a Prostate Cancer Xenograft Model.
Maddeboina K, Jonnalagadda SK, Morsy A, Duan L, Chhonker YS, Murry DJ, Penning TM, Trippier PC.
Maddeboina K, et al.
J Med Chem. 2023 Jul 27;66(14):9894-9915. doi: 10.1021/acs.jmedchem.3c00732. Epub 2023 Jul 10.
J Med Chem. 2023.
PMID: 37428858
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LC-MS/MS method for the quantitation of a dual PI3K/BRD4 inhibitor SF2523 in mouse plasma: Application to plasma protein binding and metabolism studies.
Bala V, Chhonker YS, Morales GA, Maddeboina K, Pal D, Durden DL, Murry DJ.
Bala V, et al. Among authors: maddeboina k.
Biomed Chromatogr. 2023 Aug;37(8):e5643. doi: 10.1002/bmc.5643. Epub 2023 Apr 27.
Biomed Chromatogr. 2023.
PMID: 37042063
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Facile Protocol for the Synthesis of Self-assembling Polyamine-based Peptide Amphiphiles (PPAs) and Related Biomaterials.
Samad MB, Maddeboina K, Rodrigues de Almeida N, Conda-Sheridan M.
Samad MB, et al. Among authors: maddeboina k.
J Vis Exp. 2018 Jun 25;(136):57908. doi: 10.3791/57908.
J Vis Exp. 2018.
PMID: 29985361
Free PMC article.
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Discovery of an Aldo-Keto reductase 1C3 (AKR1C3) degrader.
Carmona AV, Jonnalagadda S, Case AM, Maddeboina K, Jonnalagadda SK, Dow LF, Duan L, Penning TM, Trippier PC.
Carmona AV, et al. Among authors: maddeboina k.
Commun Chem. 2024 Apr 29;7(1):95. doi: 10.1038/s42004-024-01177-4.
Commun Chem. 2024.
PMID: 38684887
Free PMC article.
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Recent advances in multitarget-directed ligands via in silico drug discovery.
Maddeboina K, Yada B, Kumari S, McHale C, Pal D, Durden DL.
Maddeboina K, et al.
Drug Discov Today. 2024 Mar;29(3):103904. doi: 10.1016/j.drudis.2024.103904. Epub 2024 Jan 26.
Drug Discov Today. 2024.
PMID: 38280625
Review.
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