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Inhibitors of ApiAP2 protein DNA binding exhibit multistage activity against Plasmodium parasites.
PLoS Pathog. 2022 Oct 12;18(10):e1010887. doi: 10.1371/journal.ppat.1010887. eCollection 2022 Oct.
PLoS Pathog. 2022.
PMID: 36223427
Free PMC article.
Identification and genome-wide prediction of DNA binding specificities for the ApiAP2 family of regulators from the malaria parasite.
Campbell TL, De Silva EK, Olszewski KL, Elemento O, Llinás M.
Campbell TL, et al. Among authors: de silva ek.
PLoS Pathog. 2010 Oct 28;6(10):e1001165. doi: 10.1371/journal.ppat.1001165.
PLoS Pathog. 2010.
PMID: 21060817
Free PMC article.
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Structural determinants of DNA binding by a P. falciparum ApiAP2 transcriptional regulator.
Lindner SE, De Silva EK, Keck JL, Llinás M.
Lindner SE, et al. Among authors: de silva ek.
J Mol Biol. 2010 Jan 22;395(3):558-67. doi: 10.1016/j.jmb.2009.11.004. Epub 2009 Nov 10.
J Mol Biol. 2010.
PMID: 19913037
Free PMC article.
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Specific DNA-binding by apicomplexan AP2 transcription factors.
De Silva EK, Gehrke AR, Olszewski K, León I, Chahal JS, Bulyk ML, Llinás M.
De Silva EK, et al.
Proc Natl Acad Sci U S A. 2008 Jun 17;105(24):8393-8. doi: 10.1073/pnas.0801993105. Epub 2008 Jun 9.
Proc Natl Acad Sci U S A. 2008.
PMID: 18541913
Free PMC article.
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ApiAP2 transcription factor restricts development of the Toxoplasma tissue cyst.
Radke JB, Lucas O, De Silva EK, Ma Y, Sullivan WJ Jr, Weiss LM, Llinas M, White MW.
Radke JB, et al. Among authors: de silva ek.
Proc Natl Acad Sci U S A. 2013 Apr 23;110(17):6871-6. doi: 10.1073/pnas.1300059110. Epub 2013 Apr 9.
Proc Natl Acad Sci U S A. 2013.
PMID: 23572590
Free PMC article.
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A triplex-forming sequence from the human c-MYC promoter interferes with DNA transcription.
Belotserkovskii BP, De Silva E, Tornaletti S, Wang G, Vasquez KM, Hanawalt PC.
Belotserkovskii BP, et al.
J Biol Chem. 2007 Nov 2;282(44):32433-41. doi: 10.1074/jbc.M704618200. Epub 2007 Sep 4.
J Biol Chem. 2007.
PMID: 17785457
Free article.
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