Lherbet C - Search Results

1

Isoniazid Linked to Sulfonate Esters via Hydrazone Functionality: Design, Synthesis, and Evaluation of Antitubercular Activity.

Koçak Aslan E, Han Mİ, Krishna VS, Tamhaev R, Dengiz C, Doğan ŞD, Lherbet C, Mourey L, Tønjum T, Gündüz MG. Koçak Aslan E, et al. Among authors: lherbet c. Pharmaceuticals (Basel). 2022 Oct 21;15(10):1301. doi: 10.3390/ph15101301. Pharmaceuticals (Basel). 2022. PMID: 36297413 Free PMC article.

2

Expression, purification, crystallization and preliminary crystallographic analysis of Trypanosoma brucei phosphofructokinase.

Keillor JW, Lherbet C, Castonguay R, Lapierre D, Martinez-Oyanedel J, Fothergill-Gilmore LA, Walkinshaw MD. Keillor JW, et al. Among authors: lherbet c. Acta Crystallogr D Biol Crystallogr. 2003 Mar;59(Pt 3):532-4. doi: 10.1107/s0907444902023478. Epub 2003 Feb 21. Acta Crystallogr D Biol Crystallogr. 2003. PMID: 12595717

3

Crystal structure of the enoyl-ACP reductase of Mycobacterium tuberculosis (InhA) in the apo-form and in complex with the active metabolite of isoniazid pre-formed by a biomimetic approach.

Chollet A, Mourey L, Lherbet C, Delbot A, Julien S, Baltas M, Bernadou J, Pratviel G, Maveyraud L, Bernardes-Génisson V. Chollet A, et al. Among authors: lherbet c. J Struct Biol. 2015 Jun;190(3):328-37. doi: 10.1016/j.jsb.2015.04.008. Epub 2015 Apr 17. J Struct Biol. 2015. PMID: 25891098

4

Insights into Substrate Modification by Dehydratases from Type I Polyketide Synthases.

Faille A, Gavalda S, Slama N, Lherbet C, Maveyraud L, Guillet V, Laval F, Quémard A, Mourey L, Pedelacq JD. Faille A, et al. Among authors: lherbet c. J Mol Biol. 2017 May 19;429(10):1554-1569. doi: 10.1016/j.jmb.2017.03.026. Epub 2017 Apr 1. J Mol Biol. 2017. PMID: 28377293

5

Mechanochemical Synthesis and Biological Evaluation of Novel Isoniazid Derivatives with Potent Antitubercular Activity.

Oliveira PFM, Guidetti B, Chamayou A, André-Barrès C, Madacki J, Korduláková J, Mori G, Orena BS, Chiarelli LR, Pasca MR, Lherbet C, Carayon C, Massou S, Baron M, Baltas M. Oliveira PFM, et al. Among authors: lherbet c. Molecules. 2017 Sep 1;22(9):1457. doi: 10.3390/molecules22091457. Molecules. 2017. PMID: 28862683 Free PMC article.

6

Discovery of hydrazone containing thiadiazoles as Mycobacterium tuberculosis growth and enoyl acyl carrier protein reductase (InhA) inhibitors.

Doğan H, Doğan ŞD, Gündüz MG, Krishna VS, Lherbet C, Sriram D, Şahin O, Sarıpınar E. Doğan H, et al. Among authors: lherbet c. Eur J Med Chem. 2020 Feb 15;188:112035. doi: 10.1016/j.ejmech.2020.112035. Epub 2020 Jan 7. Eur J Med Chem. 2020. PMID: 31951850

7

Design and synthesis of thiourea-based derivatives as Mycobacterium tuberculosis growth and enoyl acyl carrier protein reductase (InhA) inhibitors.

Doğan ŞD, Gündüz MG, Doğan H, Krishna VS, Lherbet C, Sriram D. Doğan ŞD, et al. Among authors: lherbet c. Eur J Med Chem. 2020 Aug 1;199:112402. doi: 10.1016/j.ejmech.2020.112402. Epub 2020 May 4. Eur J Med Chem. 2020. PMID: 32417538

8

Urea derivatives carrying a thiophenylthiazole moiety: Design, synthesis, and evaluation of antitubercular and InhA inhibitory activities.

Keleş Atıcı R, Doğan ŞD, Gündüz MG, Krishna VS, Chebaiki M, Homberset H, Lherbet C, Mourey L, Tønjum T. Keleş Atıcı R, et al. Among authors: lherbet c. Drug Dev Res. 2022 Sep;83(6):1292-1304. doi: 10.1002/ddr.21958. Epub 2022 Jun 29. Drug Dev Res. 2022. PMID: 35769019

9

Discovery of new diaryl ether inhibitors against Mycobacterium tuberculosis targeting the minor portal of InhA.

Chebaiki M, Delfourne E, Tamhaev R, Danoun S, Rodriguez F, Hoffmann P, Grosjean E, Goncalves F, Azéma-Despeyroux J, Pál A, Korduláková J, Preuilh N, Britton S, Constant P, Marrakchi H, Maveyraud L, Mourey L, Lherbet C. Chebaiki M, et al. Among authors: lherbet c. Eur J Med Chem. 2023 Nov 5;259:115646. doi: 10.1016/j.ejmech.2023.115646. Epub 2023 Jul 16. Eur J Med Chem. 2023. PMID: 37482022

10

Exploring the plasticity of the InhA substrate-binding site using new diaryl ether inhibitors.

Tamhaev R, Grosjean E, Ahamed H, Chebaiki M, Rodriguez F, Recchia D, Degiacomi G, Pasca MR, Maveyraud L, Mourey L, Lherbet C. Tamhaev R, et al. Among authors: lherbet c. Bioorg Chem. 2024 Feb;143:107032. doi: 10.1016/j.bioorg.2023.107032. Epub 2023 Dec 12. Bioorg Chem. 2024. PMID: 38128204

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