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Migration mediated by the oxysterol receptor GPR183 depends on arrestin coupling but not receptor internalization.
Sci Signal. 2023 Apr 4;16(779):eabl4283. doi: 10.1126/scisignal.abl4283. Epub 2023 Apr 4.
Sci Signal. 2023.
PMID: 37014928
Discovery of GPR183 Agonists Based on an Antagonist Scaffold.
Kjaer VMS, Ieremias L, Daugvilaite V, Lückmann M, Frimurer TM, Ulven T, Rosenkilde MM, Våbenø J.
Kjaer VMS, et al.
ChemMedChem. 2021 Sep 6;16(17):2623-2627. doi: 10.1002/cmdc.202100301. Epub 2021 Aug 3.
ChemMedChem. 2021.
PMID: 34270165
Free PMC article.
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Ligand entry pathways control the chemical space recognized by GPR183.
Kjær VMS, Stępniewski TM, Medel-Lacruz B, Reinmuth L, Ciba M, Rexen Ulven E, Bonomi M, Selent J, Rosenkilde MM.
Kjær VMS, et al.
Chem Sci. 2023 Sep 25;14(39):10671-10683. doi: 10.1039/d2sc05962b. eCollection 2023 Oct 11.
Chem Sci. 2023.
PMID: 37829039
Free PMC article.
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GPR183 Is Dispensable for B1 Cell Accumulation and Function, but Affects B2 Cell Abundance, in the Omentum and Peritoneal Cavity.
Barington L, Christensen LVV, Pedersen KK, Niss Arfelt K, Roumain M, Jensen KHR, Kjær VMS, Daugvilaite V, Kearney JF, Christensen JP, Hjortø GM, Muccioli GG, Holst PJ, Rosenkilde MM.
Barington L, et al. Among authors: kjaer vms.
Cells. 2022 Jan 31;11(3):494. doi: 10.3390/cells11030494.
Cells. 2022.
PMID: 35159303
Free PMC article.
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