Gavriil ES - Search Results

1

Design, Synthesis, and Evaluation of Inhibitors of Hedgehog Acyltransferase.

Ritzefeld M, Zhang L, Xiao Z, Andrei SA, Boyd O, Masumoto N, Rodgers UR, Artelsmair M, Sefer L, Hayes A, Gavriil ES, Raynaud FI, Burke R, Blagg J, Rzepa HS, Siebold C, Magee AI, Lanyon-Hogg T, Tate EW. Ritzefeld M, et al. Among authors: gavriil es. J Med Chem. 2024 Jan 25;67(2):1061-1078. doi: 10.1021/acs.jmedchem.3c01363. Epub 2024 Jan 10. J Med Chem. 2024. PMID: 38198226 Free PMC article.

2

Design, synthesis and biological evaluation of novel substituted purine isosters as EGFR kinase inhibitors, with promising pharmacokinetic profile and in vivo efficacy.

Gavriil ES, Doukatas A, Karampelas T, Myrianthopoulos V, Dimitrakis S, Mikros E, Marakos P, Tamvakopoulos C, Pouli N. Gavriil ES, et al. Eur J Med Chem. 2019 Aug 15;176:393-409. doi: 10.1016/j.ejmech.2019.05.029. Epub 2019 May 8. Eur J Med Chem. 2019. PMID: 31125894

3

Design and synthesis of purine analogues as highly specific ligands for FcyB, a ubiquitous fungal nucleobase transporter.

Lougiakis N, Gavriil ES, Kairis M, Sioupouli G, Lambrinidis G, Benaki D, Krypotou E, Mikros E, Marakos P, Pouli N, Diallinas G. Lougiakis N, et al. Among authors: gavriil es. Bioorg Med Chem. 2016 Nov 15;24(22):5941-5952. doi: 10.1016/j.bmc.2016.09.055. Epub 2016 Sep 22. Bioorg Med Chem. 2016. PMID: 27720327

4

Structure-activity relationships in fungal nucleobases transporters as dissected by the inhibitory effects of novel purine analogues.

Gavriil ES, Dimitrakis S, Papadaki G, Balaska S, Lambrinidis G, Lougiakis N, Marakos P, Diallinas G, Pouli N, Mikros E. Gavriil ES, et al. Eur J Med Chem. 2018 Aug 5;156:240-251. doi: 10.1016/j.ejmech.2018.06.038. Epub 2018 Jun 18. Eur J Med Chem. 2018. PMID: 30006169

5

Synthesis and antiproliferative activity of new pyrazolo[3,4-c]pyridines.

Gavriil ES, Lougiakis N, Pouli N, Marakos P, Skaltsounis AL, Nam S, Jove R, Horne D, Gioti K, Pratsinis H, Kletsas D, Tenta R. Gavriil ES, et al. Med Chem. 2016 Dec 13. Online ahead of print. Med Chem. 2016. PMID: 27978787

6

Novel Substituted Purine Isosteres: Synthesis, Structure-Activity Relationships and Cytotoxic Activity Evaluation.

Dimitrakis S, Gavriil ES, Pousias A, Lougiakis N, Marakos P, Pouli N, Gioti K, Tenta R. Dimitrakis S, et al. Among authors: gavriil es. Molecules. 2021 Dec 31;27(1):247. doi: 10.3390/molecules27010247. Molecules. 2021. PMID: 35011476 Free PMC article.

7

Tat mediates apoptosis in vivo in the rat central nervous system.

Gavriil ES, Cooney R, Weeks BS. Gavriil ES, et al. Biochem Biophys Res Commun. 2000 Jan 7;267(1):252-6. doi: 10.1006/bbrc.1999.1894. Biochem Biophys Res Commun. 2000. PMID: 10623606

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