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Antascomicin B stabilizes FKBP51-Akt1 complexes as a molecular glue.
Bioorg Med Chem Lett. 2024 May 15;104:129728. doi: 10.1016/j.bmcl.2024.129728. Epub 2024 Apr 4.
Bioorg Med Chem Lett. 2024.
PMID: 38582133
Free article.
Structure-Based Design of High-Affinity Macrocyclic FKBP51 Inhibitors.
Bauder M, Meyners C, Purder PL, Merz S, Sugiarto WO, Voll AM, Heymann T, Hausch F.
Bauder M, et al. Among authors: voll am.
J Med Chem. 2021 Mar 25;64(6):3320-3349. doi: 10.1021/acs.jmedchem.0c02195. Epub 2021 Mar 5.
J Med Chem. 2021.
PMID: 33666419
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Macrocyclic FKBP51 Ligands Define a Transient Binding Mode with Enhanced Selectivity.
Voll AM, Meyners C, Taubert MC, Bajaj T, Heymann T, Merz S, Charalampidou A, Kolos J, Purder PL, Geiger TM, Wessig P, Gassen NC, Bracher A, Hausch F.
Voll AM, et al.
Angew Chem Int Ed Engl. 2021 Jun 7;60(24):13257-13263. doi: 10.1002/anie.202017352. Epub 2021 May 7.
Angew Chem Int Ed Engl. 2021.
PMID: 33843131
Free PMC article.
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FKBP Ligands-Where We Are and Where to Go?
Kolos JM, Voll AM, Bauder M, Hausch F.
Kolos JM, et al. Among authors: voll am.
Front Pharmacol. 2018 Dec 5;9:1425. doi: 10.3389/fphar.2018.01425. eCollection 2018.
Front Pharmacol. 2018.
PMID: 30568592
Free PMC article.
Review.
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The selective FKBP51 inhibitor SAFit2 reduces alcohol consumption and reinstatement of conditioned alcohol effects in mice.
König L, Kalinichenko LS, Huber SE, Voll AM, Bauder M, Kornhuber J, Hausch F, Müller CP.
König L, et al. Among authors: voll am.
Addict Biol. 2020 May;25(3):e12758. doi: 10.1111/adb.12758. Epub 2019 Jun 7.
Addict Biol. 2020.
PMID: 31173432
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Picomolar FKBP inhibitors enabled by a single water-displacing methyl group in bicyclic [4.3.1] aza-amides.
Kolos JM, Pomplun S, Jung S, Rieß B, Purder PL, Voll AM, Merz S, Gnatzy M, Geiger TM, Quist-Løkken I, Jatzlau J, Knaus P, Holien T, Bracher A, Meyners C, Czodrowski P, Krewald V, Hausch F.
Kolos JM, et al. Among authors: voll am.
Chem Sci. 2021 Nov 3;12(44):14758-14765. doi: 10.1039/d1sc04638a. eCollection 2021 Nov 17.
Chem Sci. 2021.
PMID: 34820091
Free PMC article.
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Structural and Dynamical Basis of G Protein Inhibition by YM-254890 and FR900359: An Inhibitor in Action.
Tietze D, Kaufmann D, Tietze AA, Voll A, Reher R, König G, Hausch F.
Tietze D, et al.
J Chem Inf Model. 2019 Oct 28;59(10):4361-4373. doi: 10.1021/acs.jcim.9b00433. Epub 2019 Sep 26.
J Chem Inf Model. 2019.
PMID: 31539242
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