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Conformational and Electronic Variations in 1,2- and 1,5a-Cyclophellitols and their Impact on Retaining α-Glucosidase Inhibition.
Ofman TP, Heming JJA, Nin-Hill A, Küllmer F, Moran E, Bennett M, Steneker R, Klein AM, Ruijgrok G, Kok K, Armstrong ZWB, Aerts JMFG, van der Marel GA, Rovira C, Davies GJ, Artola M, Codée JDC, Overkleeft HS. Ofman TP, et al. Among authors: artola m. Chemistry. 2024 Jun 3;30(31):e202400723. doi: 10.1002/chem.202400723. Epub 2024 Apr 24. Chemistry. 2024. PMID: 38623783
Carba-cyclophellitols Are Neutral Retaining-Glucosidase Inhibitors.
Beenakker TJM, Wander DPA, Offen WA, Artola M, Raich L, Ferraz MJ, Li KY, Houben JHPM, van Rijssel ER, Hansen T, van der Marel GA, Codée JDC, Aerts JMFG, Rovira C, Davies GJ, Overkleeft HS. Beenakker TJM, et al. Among authors: artola m. J Am Chem Soc. 2017 May 17;139(19):6534-6537. doi: 10.1021/jacs.7b01773. Epub 2017 May 5. J Am Chem Soc. 2017. PMID: 28463498 Free PMC article.
1,6-Cyclophellitol Cyclosulfates: A New Class of Irreversible Glycosidase Inhibitor.
Artola M, Wu L, Ferraz MJ, Kuo CL, Raich L, Breen IZ, Offen WA, Codée JDC, van der Marel GA, Rovira C, Aerts JMFG, Davies GJ, Overkleeft HS. Artola M, et al. ACS Cent Sci. 2017 Jul 26;3(7):784-793. doi: 10.1021/acscentsci.7b00214. Epub 2017 Jul 13. ACS Cent Sci. 2017. PMID: 28776021 Free PMC article.
Gluco-1 H-imidazole: A New Class of Azole-Type β-Glucosidase Inhibitor.
Schröder SP, Wu L, Artola M, Hansen T, Offen WA, Ferraz MJ, Li KY, Aerts JMFG, van der Marel GA, Codée JDC, Davies GJ, Overkleeft HS. Schröder SP, et al. Among authors: artola m. J Am Chem Soc. 2018 Apr 18;140(15):5045-5048. doi: 10.1021/jacs.8b02399. Epub 2018 Apr 4. J Am Chem Soc. 2018. PMID: 29601200 Free PMC article.
New Irreversible α-l-Iduronidase Inhibitors and Activity-Based Probes.
Artola M, Kuo CL, McMahon SA, Oehler V, Hansen T, van der Lienden M, He X, van den Elst H, Florea BI, Kermode AR, van der Marel GA, Gloster TM, Codée JDC, Overkleeft HS, Aerts JMFG. Artola M, et al. Chemistry. 2018 Dec 17;24(71):19081-19088. doi: 10.1002/chem.201804662. Epub 2018 Nov 26. Chemistry. 2018. PMID: 30307091 Free PMC article.
Rational Design of Mechanism-Based Inhibitors and Activity-Based Probes for the Identification of Retaining α-l-Arabinofuranosidases.
McGregor NGS, Artola M, Nin-Hill A, Linzel D, Haon M, Reijngoud J, Ram A, Rosso MN, van der Marel GA, Codée JDC, van Wezel GP, Berrin JG, Rovira C, Overkleeft HS, Davies GJ. McGregor NGS, et al. Among authors: artola m. J Am Chem Soc. 2020 Mar 11;142(10):4648-4662. doi: 10.1021/jacs.9b11351. Epub 2020 Feb 26. J Am Chem Soc. 2020. PMID: 32053363 Free PMC article.
Design, Synthesis and Structural Analysis of Glucocerebrosidase Imaging Agents.
Rowland RJ, Chen Y, Breen I, Wu L, Offen WA, Beenakker TJ, Su Q, van den Nieuwendijk AMCH, Aerts JMFG, Artola M, Overkleeft HS, Davies GJ. Rowland RJ, et al. Among authors: artola m. Chemistry. 2021 Nov 25;27(66):16377-16388. doi: 10.1002/chem.202102359. Epub 2021 Oct 29. Chemistry. 2021. PMID: 34570911 Free PMC article.
1,6-epi-Cyclophellitol Cyclosulfamidate Is a Bona Fide Lysosomal α-Glucosidase Stabilizer for the Treatment of Pompe Disease.
Kok K, Kuo CL, Katzy RE, Lelieveld LT, Wu L, Roig-Zamboni V, van der Marel GA, Codée JDC, Sulzenbacher G, Davies GJ, Overkleeft HS, Aerts JMFG, Artola M. Kok K, et al. Among authors: artola m. J Am Chem Soc. 2022 Aug 17;144(32):14819-14827. doi: 10.1021/jacs.2c05666. Epub 2022 Aug 2. J Am Chem Soc. 2022. PMID: 35917590 Free PMC article.
63 results