R01 AI087671/AI/NIAID NIH HHS/United States[Grants and Funding] - Search Results

Year	Number of Results
2010	1
2011	3
2012	2
2013	3
2014	6
2015	3
2016	5
2017	1
2018	4
2019	3
2020	1
2023	1
2024	0

1

Delgado JL, Hsieh CM, Chan NL, Hiasa H. Delgado JL, et al. Biochem J. 2018 Jan 23;475(2):373-398. doi: 10.1042/BCJ20160583. Biochem J. 2018. PMID: 29363591 Free PMC article. Review.

2

Mechanism of quinolone action and resistance.

Aldred KJ, Kerns RJ, Osheroff N. Aldred KJ, et al. Biochemistry. 2014 Mar 18;53(10):1565-74. doi: 10.1021/bi5000564. Epub 2014 Mar 7. Biochemistry. 2014. PMID: 24576155 Free PMC article. Review.

3

DNA Topoisomerases as Targets for Antibacterial Agents.

Hiasa H. Hiasa H. Methods Mol Biol. 2018;1703:47-62. doi: 10.1007/978-1-4939-7459-7_3. Methods Mol Biol. 2018. PMID: 29177732

4

Identification of an ethyl 5,6-dihydropyrazolo[1,5-c]quinazoline-1-carboxylate as a catalytic inhibitor of DNA gyrase.

Aguirre AL, Chheda PR, Lentz SRC, Held HA, Groves NP, Hiasa H, Kerns RJ. Aguirre AL, et al. Bioorg Med Chem. 2020 May 15;28(10):115439. doi: 10.1016/j.bmc.2020.115439. Epub 2020 Mar 13. Bioorg Med Chem. 2020. PMID: 32234278 Free PMC article.

5

Suppression of gyrase-mediated resistance by C7 aryl fluoroquinolones.

Malik M, Mustaev A, Schwanz HA, Luan G, Shah N, Oppegard LM, de Souza EC, Hiasa H, Zhao X, Kerns RJ, Drlica K. Malik M, et al. Nucleic Acids Res. 2016 Apr 20;44(7):3304-16. doi: 10.1093/nar/gkw161. Epub 2016 Mar 16. Nucleic Acids Res. 2016. PMID: 26984528 Free PMC article.

6

Probing structural requirements for human topoisomerase I inhibition by a novel N1-Biphenyl fluoroquinolone.

Delgado JL, Lentz SRC, Kulkarni CA, Chheda PR, Held HA, Hiasa H, Kerns RJ. Delgado JL, et al. Eur J Med Chem. 2019 Jun 15;172:109-130. doi: 10.1016/j.ejmech.2019.03.040. Epub 2019 Mar 20. Eur J Med Chem. 2019. PMID: 30959322 Free PMC article.

7

Fluoroquinolone-gyrase-DNA complexes: two modes of drug binding.

Mustaev A, Malik M, Zhao X, Kurepina N, Luan G, Oppegard LM, Hiasa H, Marks KR, Kerns RJ, Berger JM, Drlica K. Mustaev A, et al. J Biol Chem. 2014 May 2;289(18):12300-12. doi: 10.1074/jbc.M113.529164. Epub 2014 Feb 4. J Biol Chem. 2014. PMID: 24497635 Free PMC article.

8

The C7-aminomethylpyrrolidine group rescues the activity of a thio-fluoroquinolone.

Lentz SRC, Chheda PR, Oppegard LM, Towle TR, Kerns RJ, Hiasa H. Lentz SRC, et al. Biochimie. 2019 May;160:24-27. doi: 10.1016/j.biochi.2019.02.002. Epub 2019 Feb 11. Biochimie. 2019. PMID: 30763638 Free PMC article.

9

Resveratrol Antagonizes Antimicrobial Lethality and Stimulates Recovery of Bacterial Mutants.

Liu Y, Zhou J, Qu Y, Yang X, Shi G, Wang X, Hong Y, Drlica K, Zhao X. Liu Y, et al. PLoS One. 2016 Apr 5;11(4):e0153023. doi: 10.1371/journal.pone.0153023. eCollection 2016. PLoS One. 2016. PMID: 27045517 Free PMC article.

10

Role of the Water-Metal Ion Bridge in Quinolone Interactions with Escherichia coli Gyrase.

Carter HE, Wildman B, Schwanz HA, Kerns RJ, Aldred KJ. Carter HE, et al. Int J Mol Sci. 2023 Feb 2;24(3):2879. doi: 10.3390/ijms24032879. Int J Mol Sci. 2023. PMID: 36769202 Free PMC article.

Save citations to file

Email citations

Send citations to clipboard

Add to Collections

Add to My Bibliography

Create a file for external citation management software

Your saved search

Your RSS Feed

My NCBI Filters

Results by year

Text availability

Article attribute

Article type

Publication date

29 results

Results by year

Search Page

Filters

My NCBI Filters

Results by year

Text availability

Article attribute

Article type

Publication date

Search Results

29 results

Results by year