Alvarez-Builla J - Search Results

1

A novel pipeline of 2-(benzenesulfonamide)-N-(4-hydroxyphenyl) acetamide analgesics that lack hepatotoxicity and retain antipyresis.

Bazan HA, Bhattacharjee S, Burgos C, Recio J, Abet V, Pahng AR, Jun B, Heap J, Ledet AJ, Gordon WC, Edwards S, Paul D, Alvarez-Builla J, Bazan NG. Bazan HA, et al. Among authors: alvarez builla j. Eur J Med Chem. 2020 Sep 15;202:112600. doi: 10.1016/j.ejmech.2020.112600. Epub 2020 Jun 30. Eur J Med Chem. 2020. PMID: 32629335 Free PMC article.

2

Prodrug approach: An overview of recent cases.

Abet V, Filace F, Recio J, Alvarez-Builla J, Burgos C. Abet V, et al. Among authors: alvarez builla j. Eur J Med Chem. 2017 Feb 15;127:810-827. doi: 10.1016/j.ejmech.2016.10.061. Epub 2016 Oct 29. Eur J Med Chem. 2017. PMID: 27823878 Review.

3

Synthesis and in vivo evaluation of non-hepatotoxic acetaminophen analogs.

Vaccarino AL, Paul D, Mukherjee PK, Rodríguez de Turco EB, Marcheselli VL, Xu L, Trudell ML, Minguez JM, Matía MP, Sunkel C, Alvarez-Builla J, Bazan NG. Vaccarino AL, et al. Bioorg Med Chem. 2007 Mar 1;15(5):2206-15. doi: 10.1016/j.bmc.2006.07.054. Epub 2006 Aug 21. Bioorg Med Chem. 2007. PMID: 16919959 Free article.

4

Benzo[f]azino[2,1-a]phthalazinium cations: novel DNA intercalating chromophores with antiproliferative activity.

Martínez V, Burgos C, Alvarez-Builla J, Fernández G, Domingo A, García-Nieto R, Gago F, Manzanares I, Cuevas C, Vaquero JJ. Martínez V, et al. J Med Chem. 2004 Feb 26;47(5):1136-48. doi: 10.1021/jm0310434. J Med Chem. 2004. PMID: 14971893

5

Unusual approach to 3-aryl-2-aminopyridines through a radical mechanism: synthesis and theoretical rationale from quantum mechanical calculations.

Camacho-Artacho M, Abet V, Frutos LM, Gago F, Alvarez-Builla J, Burgos C. Camacho-Artacho M, et al. J Org Chem. 2011 Mar 4;76(5):1452-5. doi: 10.1021/jo102122h. Epub 2011 Jan 25. J Org Chem. 2011. PMID: 21265527

6

Synthesis and evaluation of quinazoline derivatives as phosphodiesterase 7 inhibitors.

Sánchez AI, Martínez-Barrasa V, Burgos C, Vaquero JJ, Alvarez-Builla J, Terricabras E, Segarra V. Sánchez AI, et al. Bioorg Med Chem. 2013 Apr 15;21(8):2370-2378. doi: 10.1016/j.bmc.2013.01.067. Epub 2013 Feb 5. Bioorg Med Chem. 2013. PMID: 23454131

7

LAU-0901, a novel platelet-activating factor antagonist, is highly neuroprotective in cerebral ischemia.

Belayev L, Khoutorova L, Atkins K, Gordon WC, Alvarez-Builla J, Bazan NG. Belayev L, et al. Exp Neurol. 2008 Dec;214(2):253-8. doi: 10.1016/j.expneurol.2008.08.009. Epub 2008 Aug 28. Exp Neurol. 2008. PMID: 18793637 Free PMC article.

8

A new class of pyrazolopyridine nucleus with fluorescent properties, obtained through either a radical or a Pd arylation pathway from N-azinylpyridinium N-aminides.

Abet V, Nuñez A, Mendicuti F, Burgos C, Alvarez-Builla J. Abet V, et al. J Org Chem. 2008 Nov 21;73(22):8800-7. doi: 10.1021/jo801549u. Epub 2008 Oct 21. J Org Chem. 2008. PMID: 18937415

9

N-(4-[(18)F]-fluoropyridin-2-yl)-N-{2-[4-(2-methoxyphenyl)piperazin-1-yl]ethyl}carboxamides as analogs of WAY100635. New PET tracers of serotonin 5-HT(1A) receptors.

García G, Abet V, Alajarín R, Álvarez-Builla J, Delgado M, García-García L, Bascuñana-Almarcha P, Peña-Salcedo C, Kelly J, Pozo MA. García G, et al. Among authors: alvarez builla j. Eur J Med Chem. 2014 Oct 6;85:795-806. doi: 10.1016/j.ejmech.2014.07.096. Epub 2014 Jul 26. Eur J Med Chem. 2014. PMID: 25171752

10

DNA sequence-specific reading by echinomycin: role of hydrogen bonding and stacking interactions.

Gallego J, Luque FJ, Orozco M, Burgos C, Alvarez-Builla J, Rodrigo MM, Gago F. Gallego J, et al. J Med Chem. 1994 May 27;37(11):1602-9. doi: 10.1021/jm00037a010. J Med Chem. 1994. PMID: 8201593

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