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Amide Bond Bioisosteres: Strategies, Synthesis, and Successes.
J Med Chem. 2020 Nov 12;63(21):12290-12358. doi: 10.1021/acs.jmedchem.0c00530. Epub 2020 Aug 4.
J Med Chem. 2020.
PMID: 32686940
Free PMC article.
Review.
Exogenous Flupirtine as Potential Treatment for CLN3 Disease.
Maalouf K, Makoukji J, Saab S, Makhoul NJ, Carmona AV, Kinarivala N, Ghanem N, Trippier PC, Boustany RM.
Maalouf K, et al. Among authors: carmona av.
Cells. 2020 Aug 11;9(8):1872. doi: 10.3390/cells9081872.
Cells. 2020.
PMID: 32796515
Free PMC article.
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An iPSC-Derived Neuron Model of CLN3 Disease Facilitates Small Molecule Phenotypic Screening.
Kinarivala N, Morsy A, Patel R, Carmona AV, Sajib MS, Raut S, Mikelis CM, Al-Ahmad A, Trippier PC.
Kinarivala N, et al. Among authors: carmona av.
ACS Pharmacol Transl Sci. 2020 Sep 1;3(5):931-947. doi: 10.1021/acsptsci.0c00077. eCollection 2020 Oct 9.
ACS Pharmacol Transl Sci. 2020.
PMID: 33073192
Free PMC article.
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Patient-Derived Induced Pluripotent Stem Cell Models for Phenotypic Screening in the Neuronal Ceroid Lipofuscinoses.
Morsy A, Carmona AV, Trippier PC.
Morsy A, et al. Among authors: carmona av.
Molecules. 2021 Oct 15;26(20):6235. doi: 10.3390/molecules26206235.
Molecules. 2021.
PMID: 34684815
Free PMC article.
Review.
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Discovery of an Aldo-Keto reductase 1C3 (AKR1C3) degrader.
Carmona AV, Jonnalagadda S, Case AM, Maddeboina K, Jonnalagadda SK, Dow LF, Duan L, Penning TM, Trippier PC.
Carmona AV, et al.
Commun Chem. 2024 Apr 29;7(1):95. doi: 10.1038/s42004-024-01177-4.
Commun Chem. 2024.
PMID: 38684887
Free PMC article.
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