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A new class of cytotoxic agents targets tubulin and disrupts microtubule dynamics.
Bioorg Chem. 2021 Nov;116:105297. doi: 10.1016/j.bioorg.2021.105297. Epub 2021 Aug 30.
Bioorg Chem. 2021.
PMID: 34509798
Free PMC article.
The structural requirements of histone deacetylase inhibitors: C4-modified SAHA analogs display dual HDAC6/HDAC8 selectivity.
Negmeldin AT, Knoff JR, Pflum MKH.
Negmeldin AT, et al. Among authors: knoff jr.
Eur J Med Chem. 2018 Jan 1;143:1790-1806. doi: 10.1016/j.ejmech.2017.10.076. Epub 2017 Oct 31.
Eur J Med Chem. 2018.
PMID: 29150330
Free PMC article.
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First-in-Class Dual Mechanism Ferroptosis-HDAC Inhibitor Hybrids.
Karaj E, Sindi SH, Kuganesan N, Koranne RA, Knoff JR, James AW, Fu Y, Kotsull LN, Pflum MK, Shah Z, Taylor WR, Tillekeratne LMV.
Karaj E, et al. Among authors: knoff jr.
J Med Chem. 2022 Nov 10;65(21):14764-14791. doi: 10.1021/acs.jmedchem.2c01276. Epub 2022 Oct 28.
J Med Chem. 2022.
PMID: 36306372
Free PMC article.
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