Hlasta DJ - Search Results

1

2,6-Disubstituted aryl carboxylic acids, leaving groups "par excellence" for benzisothiazolone inhibitors of human leukocyte elastase.

Subramanyam C, Bell MR, Carabateas P, Court JJ, Dority JA Jr, Ferguson E, Gordon R, Hlasta DJ, Kumar V, Saindane M, et al. Subramanyam C, et al. Among authors: hlasta dj. J Med Chem. 1994 Aug 19;37(17):2623-6. doi: 10.1021/jm00043a001. J Med Chem. 1994. PMID: 8064791 No abstract available.

2

5-Lipoxygenase inhibitors: the synthesis and structure-activity relationships of a series of 1-phenyl-3-pyrazolidinones.

Hlasta DJ, Casey FB, Ferguson EW, Gangell SJ, Heimann MR, Jaeger EP, Kullnig RK, Gordon RJ. Hlasta DJ, et al. J Med Chem. 1991 May;34(5):1560-70. doi: 10.1021/jm00109a006. J Med Chem. 1991. PMID: 1903450

3

A novel class of cyclic beta-dicarbonyl leaving groups and their use in the design of benzisothiazolone human leukocyte elastase inhibitors.

Hlasta DJ, Ackerman JH, Court JJ, Farrell RP, Johnson JA, Kofron JL, Robinson DT, Talomie TG, Dunlap RP, Franke CA. Hlasta DJ, et al. J Med Chem. 1995 Nov 10;38(23):4687-92. doi: 10.1021/jm00023a008. J Med Chem. 1995. PMID: 7473596

4

Phosphonates and phosphinates: novel leaving groups for benzisothiazolone inhibitors of human leukocyte elastase.

Desai RC, Court JC, Ferguson E, Gordon RJ, Hlasta DJ, Dunlap RP, Franke CA. Desai RC, et al. Among authors: hlasta dj. J Med Chem. 1995 Apr 28;38(9):1571-4. doi: 10.1021/jm00009a017. J Med Chem. 1995. PMID: 7739015

5

Orally bioavailable benzisothiazolone inhibitors of human leukocyte elastase.

Hlasta DJ, Subramanyam C, Bell MR, Carabateas PM, Court JJ, Desai RC, Drozd ML, Eickhoff WM, Ferguson EW, Gordon RJ, et al. Hlasta DJ, et al. J Med Chem. 1995 Mar 3;38(5):739-44. doi: 10.1021/jm00005a001. J Med Chem. 1995. PMID: 7877139

6

Antinociceptive (aminoalkyl)indoles.

Bell MR, D'Ambra TE, Kumar V, Eissenstat MA, Herrmann JL Jr, Wetzel JR, Rosi D, Philion RE, Daum SJ, Hlasta DJ, et al. Bell MR, et al. Among authors: hlasta dj. J Med Chem. 1991 Mar;34(3):1099-110. doi: 10.1021/jm00107a034. J Med Chem. 1991. PMID: 1900533

7

Substituted salicylanilides as inhibitors of two-component regulatory systems in bacteria.

Macielag MJ, Demers JP, Fraga-Spano SA, Hlasta DJ, Johnson SG, Kanojia RM, Russell RK, Sui Z, Weidner-Wells MA, Werblood H, Foleno BD, Goldschmidt RM, Loeloff MJ, Webb GC, Barrett JF. Macielag MJ, et al. Among authors: hlasta dj. J Med Chem. 1998 Jul 30;41(16):2939-45. doi: 10.1021/jm9803572. J Med Chem. 1998. PMID: 9685233

8

Synthesis and biological evaluation of novel pyridazinone-based alpha4 integrin receptor antagonists.

Gong Y, Barbay JK, Dyatkin AB, Miskowski TA, Kimball ES, Prouty SM, Fisher MC, Santulli RJ, Schneider CR, Wallace NH, Ballentine SA, Hageman WE, Masucci JA, Maryanoff BE, Damiano BP, Andrade-Gordon P, Hlasta DJ, Hornby PJ, He W. Gong Y, et al. Among authors: hlasta dj. J Med Chem. 2006 Jun 1;49(11):3402-11. doi: 10.1021/jm060031q. J Med Chem. 2006. PMID: 16722660

9

Synthesis and structure-activity relationships of 3,5-diarylisoxazoles and 3,5-diaryl-1,2,4-oxadiazoles, novel classes of small molecule interleukin-8 (IL-8) receptor antagonists.

Weidner-Wells MA, Henninger TC, Fraga-Spano SA, Boggs CM, Matheis M, Ritchie DM, Argentieri DC, Wachter MP, Hlasta DJ. Weidner-Wells MA, et al. Among authors: hlasta dj. Bioorg Med Chem Lett. 2004 Aug 16;14(16):4307-11. doi: 10.1016/j.bmcl.2004.05.080. Bioorg Med Chem Lett. 2004. PMID: 15261292

10

The synthesis and SAR of rhodanines as novel class C beta-lactamase inhibitors.

Grant EB, Guiadeen D, Baum EZ, Foleno BD, Jin H, Montenegro DA, Nelson EA, Bush K, Hlasta DJ. Grant EB, et al. Among authors: hlasta dj. Bioorg Med Chem Lett. 2000 Oct 2;10(19):2179-82. doi: 10.1016/s0960-894x(00)00444-3. Bioorg Med Chem Lett. 2000. PMID: 11012024

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